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Journal of Medicinal Chemistry|November 5, 2024
Expanding the Solvent/Protein Region Occupation of the Non-Nucleoside Reverse Transcriptase Inhibitor Binding Pocket for Improved Broad-Spectrum Anti-HIV-1 Efficacy: from Rigid Phenyl-Diarylpyrimidines to Flexible Hydrophilic Piperidine-DiarylpyrimidinesWen-Juan Huang, Christophe Pannecouque, Erik De Clercq, et al.Chemmedchem|March 30, 2026
Design and Discovery of Substituted 1,3,4-Thiadiazole-1,3,5-Triazine Hybrids as Human Immunodeficiency Virus-1 Non-Nucleoside Reverse Transcriptase Inhibitors with Anti-SARS-CoV-2 and Antibacterial ActivitiesSaumya Singh, Kumar Saurabh Srivastava, Mukesh Kumar Kumawat, et al.Frontiers in Microbiology|April 5, 2017
Chelation Motifs Affecting Metal-dependent Viral Enzymes: <i>N'</i>-acylhydrazone Ligands as Dual Target Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H DomainMauro Carcelli, Dominga Rogolino, Anna Gatti, et al.Molecules (Basel, Switzerland)|August 27, 2021
Chemical Characterization and Anti-HIV-1 Activity Assessment of Iridoids and Flavonols from <i>Scrophularia trifoliata</i>Francesca Guzzo, Rosita Russo, Cinzia Sanna, et al.Molecules (Basel, Switzerland)|May 11, 2024
Structure-Based Design of Novel Thiazolone[3,2-<i>a</i>]pyrimidine Derivatives as Potent RNase H Inhibitors for HIV TherapyXuan-De Zhu, Angela Corona, Stefania Maloccu, et al.Virulence|August 2, 2021
Zika virus NS2A inhibits interferon signaling by degradation of STAT1 and STAT2Elisa Fanunza, Fabrizio Carletti, Marina Quartu, et al.The FEBS Journal|February 26, 2011
Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and RNase H activities effective also on the RNase H activity of non-nucleoside resistant reverse transcriptasesFrancesca Esposito, Tatyana Kharlamova, Simona Distinto, et al.Pathogens and Disease|September 2, 2017
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and RDDP functionsAngela Corona, Valentina Onnis, Alessandro Deplano, et al.Polymers|June 10, 2023
Visible Light-Mediated Inactivation of H1N1 Virus UsingPolymer-Based Heterojunction PhotocatalystStefania Porcu, Stefania Maloccu, Angela Corona, et al.Viruses|December 28, 2021
INMI1 Zika Virus NS4B Antagonizes the Interferon Signaling by Suppressing STAT1 PhosphorylationElisa Fanunza, Nicole Grandi, Marina Quartu, et al.Pageof 12