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Chembiochem : a European Journal of Chemical Biology|March 7, 2016
Inhibition of HIV-1 Reverse Transcriptase Dimerization by Small MoleculesCristina Tintori, Angela Corona, Francesca Esposito, et al.Journal of Medicinal Chemistry|April 5, 2025
Deuteration Strategy-Inspired Design of Novel Diarylpyrimidine Derivatives as Potent Non-Nucleoside Reverse Transcriptase Inhibitors Featuring Improved Efficacy, Selectivity, and DruggabilityKun Zhang, Tianhao Xing, Li Ding, et al.European Journal of Medicinal Chemistry|July 5, 2014
Antiretroviral activity of metal-chelating HIV-1 integrase inhibitorsMauro Carcelli, Dominga Rogolino, Mario Sechi, et al.Molecules (Basel, Switzerland)|February 13, 2025
Identification of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Inhibitors Based on 2-Hydroxy-1,4-naphthoquinone Mannich BasesNhat Quang Tu, Clémence Richetta, Federica Putzu, et al.Molecules (Basel, Switzerland)|March 11, 2020
1,2,4-Triazolo[1,5-<i>a</i>]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H ActivityJenny Desantis, Serena Massari, Angela Corona, et al.Molecules (Basel, Switzerland)|July 15, 2026
Structure-Activity Relationships of Pyrrolyl-Containing Diketo Acid and Non-Diketo Acid Derivatives as Inhibitors of SARS-CoV-2 nsp13-Associated ActivitiesElisa Patacchini, Francesco Saccoliti, Roberta Emmolo, et al.International Journal of Molecular Sciences|August 25, 2016
Inhibitory Effect of 2,3,5,6-Tetrafluoro-4-[4-(aryl)-1H-1,2,3-triazol-1-yl]benzenesulfonamide Derivatives on HIV Reverse Transcriptase Associated RNase H ActivitiesNicolino Pala, Francesca Esposito, Dominga Rogolino, et al.European Journal of Medicinal Chemistry|January 15, 2025
Structure-based discovery of novel diarylpyrimidines as potent and selective Non-Nucleoside reverse transcriptase inhibitors: From CH(CN)-Biphenyl-Diarylpyrimidines to CNNH<sub>2</sub>-Biphenyl-DiarylpyrimidinesXiao-Mei Chen, Christophe Pannecouque, Erik De Clercq, et al.Nucleic Acids Research|February 7, 2016
Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitorsAnna Schneider, Angela Corona, Imke Spöring, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|November 4, 2020
Scaffold hopping and optimisation of 3',4'-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease HGraziella Tocco, Francesca Esposito, Pierluigi Caboni, et al.Pageof 12