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Expert Opinion on Therapeutic Patents
|
December 10, 2025
Lysine demethylase (KDM) inhibitors for the treatment of cancer: a patent review (2015-present)
Federica Sarno, Mariarosaria Conte, Annamaria Muro, et al.
Biomedicines
|
June 28, 2023
Sirtuin Inhibitor Cambinol Induces Cell Differentiation and Differently Interferes with SIRT1 and 2 at the Substrate Binding Site
Deborah Giordano, Bernardina Scafuri, Luigi De Masi, et al.
Journal of Medicinal Chemistry
|
April 29, 2005
Class II (IIa)-selective histone deacetylase inhibitors. 1. Synthesis and biological evaluation of novel (aryloxopropenyl)pyrrolyl hydroxyamides
Antonello Mai, Silvio Massa, Riccardo Pezzi, et al.
Journal of Translational Medicine
|
September 15, 2023
SIRT1 activation promotes energy homeostasis and reprograms liver cancer metabolism
Benluvankar Varghese, Ugo Chianese, Lucia Capasso, et al.
Methods in Molecular Biology (Clifton, N.J.)
|
September 4, 2014
Analysis of chromatin-nuclear receptor interactions by laser-chromatin immunoprecipitation
Rosaria Benedetti, Mariarosaria Conte, Vincenzo Carafa, et al.
The International Journal of Biochemistry & Cell Biology
|
February 5, 2008
TNF-related apoptosis-inducing ligand: signalling of a 'smart' molecule
Fabio Manzo, Angela Nebbioso, Marco Miceli, et al.
Oncogene
|
February 23, 2018
The HDAC inhibitor SAHA regulates CBX2 stability via a SUMO-triggered ubiquitin-mediated pathway in leukemia
Antonella Di Costanzo, Nunzio Del Gaudio, Lidio Conte, et al.
Journal of Medicinal Chemistry
|
September 29, 2006
Synthesis and biological properties of novel, uracil-containing histone deacetylase inhibitors
Antonello Mai, Silvio Massa, Dante Rotili, et al.
The International Journal of Biochemistry & Cell Biology
|
March 6, 2014
Identification of NuRSERY, a new functional HDAC complex composed by HDAC5, GATA1, EKLF and pERK present in human erythroid cells
Lilian Varricchio, Carmela Dell'Aversana, Angela Nebbioso, et al.
Chemmedchem
|
July 27, 2018
Synthesis and Biological Evaluation of Tripartin, a Putative KDM4 Natural Product Inhibitor, and 1-Dichloromethylinden-1-ol Analogues
Lucía Guillade, Federica Sarno, Hanna Tarhonskaya, et al.
Page
of 15
Search research articles
Search
Showing results (51-60 of 144) with videos related to
Sort By:
Page
of 15
Expert Opinion on Therapeutic Patents
|
December 10, 2025
Lysine demethylase (KDM) inhibitors for the treatment of cancer: a patent review (2015-present)
Federica Sarno, Mariarosaria Conte, Annamaria Muro, et al.
Biomedicines
|
June 28, 2023
Sirtuin Inhibitor Cambinol Induces Cell Differentiation and Differently Interferes with SIRT1 and 2 at the Substrate Binding Site
Deborah Giordano, Bernardina Scafuri, Luigi De Masi, et al.
Journal of Medicinal Chemistry
|
April 29, 2005
Class II (IIa)-selective histone deacetylase inhibitors. 1. Synthesis and biological evaluation of novel (aryloxopropenyl)pyrrolyl hydroxyamides
Antonello Mai, Silvio Massa, Riccardo Pezzi, et al.
Journal of Translational Medicine
|
September 15, 2023
SIRT1 activation promotes energy homeostasis and reprograms liver cancer metabolism
Benluvankar Varghese, Ugo Chianese, Lucia Capasso, et al.
Methods in Molecular Biology (Clifton, N.J.)
|
September 4, 2014
Analysis of chromatin-nuclear receptor interactions by laser-chromatin immunoprecipitation
Rosaria Benedetti, Mariarosaria Conte, Vincenzo Carafa, et al.
The International Journal of Biochemistry & Cell Biology
|
February 5, 2008
TNF-related apoptosis-inducing ligand: signalling of a 'smart' molecule
Fabio Manzo, Angela Nebbioso, Marco Miceli, et al.
Oncogene
|
February 23, 2018
The HDAC inhibitor SAHA regulates CBX2 stability via a SUMO-triggered ubiquitin-mediated pathway in leukemia
Antonella Di Costanzo, Nunzio Del Gaudio, Lidio Conte, et al.
Journal of Medicinal Chemistry
|
September 29, 2006
Synthesis and biological properties of novel, uracil-containing histone deacetylase inhibitors
Antonello Mai, Silvio Massa, Dante Rotili, et al.
The International Journal of Biochemistry & Cell Biology
|
March 6, 2014
Identification of NuRSERY, a new functional HDAC complex composed by HDAC5, GATA1, EKLF and pERK present in human erythroid cells
Lilian Varricchio, Carmela Dell'Aversana, Angela Nebbioso, et al.
Chemmedchem
|
July 27, 2018
Synthesis and Biological Evaluation of Tripartin, a Putative KDM4 Natural Product Inhibitor, and 1-Dichloromethylinden-1-ol Analogues
Lucía Guillade, Federica Sarno, Hanna Tarhonskaya, et al.
Page
of 15