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European Journal of Medicinal Chemistry|April 24, 2023
Application of an "inhalation by design" approach to the identification and in-vitro evaluation of novel purine based PI3Kδ inhibitorsRoberta Mazzucato, Marinella Roberti, Anna Maria Capelli, et al.The Journal of Pharmacology and Experimental Therapeutics|September 3, 2010
Identification and characterization of novel NMDA receptor antagonists selective for NR2A- over NR2B-containing receptorsEzio Bettini, Anna Sava, Cristiana Griffante, et al.British Journal of Pharmacology|January 15, 2011
Stable expression and functional characterization of a human nicotinic acetylcholine receptor with α6β2 properties: discovery of selective antagonistsAnna Maria Capelli, Laura Castelletti, Yu Hua Chen, et al.Chemmedchem|March 17, 2010
Triazolyl azabicyclo[3.1.0]hexanes: A class of potent and selective dopamine D(3) receptor antagonistsGiorgio Bonanomi, Simone Braggio, Anna Maria Capelli, et al.Journal of Medicinal Chemistry|May 11, 2017
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted AnalogsAlessio Lodola, Serena Bertolini, Matteo Biagetti, et al.Bioorganic & Medicinal Chemistry Letters|November 9, 2010
Synthesis and pharmacological characterization of 5-phenyl-2-[2-(1-piperidinylcarbonyl)phenyl]-2,3-dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones: a new class of Neuropeptide S antagonistsFabrizio Micheli, Romano Di Fabio, Angelo Giacometti, et al.Journal of Medicinal Chemistry|June 22, 2024
Discovery and Optimization of Pyridazinones as PI3Kδ Selective Inhibitors for Administration by InhalationPaolo Bruno, Alessandra Micoli, Mauro Corsi, et al.Bioorganic & Medicinal Chemistry Letters|August 10, 2011
Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-aDaniele Simoni, Riccardo Rondanin, Paolo Marchetti, et al.Bioorganic & Medicinal Chemistry Letters|January 8, 2008
New fused benzazepine as selective D3 receptor antagonists. Synthesis and biological evaluation. Part 2: [g]-fused and hetero-fused systemsFabrizio Micheli, Giorgio Bonanomi, Simone Braggio, et al.Neuropharmacology|July 16, 2011
In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE)Elisabetta Perdona', Vivian J A Costantini, Michela Tessari, et al.Pageof 4