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Bioorganic & Medicinal Chemistry
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June 21, 2024
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM study
Nace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, et al.
Tuberculosis (Edinburgh, Scotland)
|
September 13, 2018
The EU approved antimalarial pyronaridine shows antitubercular activity and synergy with rifampicin, targeting RNA polymerase
Giorgia Mori, Beatrice Silvia Orena, Clara Franch, et al.
Journal of Medicinal Chemistry
|
January 12, 2023
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against <i>Acinetobacter baumannii</i> and <i>Pseudomonas aeruginosa</i>
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, et al.
Journal of Medicinal Chemistry
|
March 6, 2023
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate <i>Staphylococcus aureus</i>
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, et al.
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Search research articles
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Showing results (141-150 of 144) with videos related to
Sort By:
Page
of 15
You have reached the last page of results.
This site can display upto 144 results.
Bioorganic & Medicinal Chemistry
|
June 21, 2024
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM study
Nace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, et al.
Tuberculosis (Edinburgh, Scotland)
|
September 13, 2018
The EU approved antimalarial pyronaridine shows antitubercular activity and synergy with rifampicin, targeting RNA polymerase
Giorgia Mori, Beatrice Silvia Orena, Clara Franch, et al.
Journal of Medicinal Chemistry
|
January 12, 2023
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against <i>Acinetobacter baumannii</i> and <i>Pseudomonas aeruginosa</i>
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, et al.
Journal of Medicinal Chemistry
|
March 6, 2023
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate <i>Staphylococcus aureus</i>
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, et al.
Page
of 15