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Journal of Medicinal Chemistry|November 25, 2014
Indolylarylsulfones carrying a heterocyclic tail as very potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitorsValeria Famiglini, Giuseppe La Regina, Antonio Coluccia, et al.European Journal of Medicinal Chemistry|December 9, 2014
New 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides inhibit hepatitis C virus replication via suppression of cyclooxygenase-2Dinesh Manvar, Sveva Pelliccia, Giuseppe La Regina, et al.European Journal of Medicinal Chemistry|May 7, 2018
New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitorsGiuseppe La Regina, Ruoli Bai, Antonio Coluccia, et al.Oncogene|March 20, 2018
β-catenin knockdown promotes NHERF1-mediated survival of colorectal cancer cells: implications for a double-targeted therapyConcetta Saponaro, Sara Sergio, Antonio Coluccia, et al.Circulation Research|January 13, 2023
Toll-Like Receptor 4-Dependent Platelet-Related Thrombosis in SARS-CoV-2 InfectionRoberto Carnevale, Vittoria Cammisotto, Simona Bartimoccia, et al.Journal of Medicinal Chemistry|August 11, 2025
Ferroptosis Induction by a New Pyrrole Derivative in Triple Negative Breast Cancer and Colorectal CancerDomiziana Masci, Lele Ling, Lian Yang, et al.Journal of Medicinal Chemistry|June 12, 2026
(<i>S</i>,<i>S</i>)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-<i>N</i>-(1-oxo-1-((1-(pyridin-4-yl)ethyl)amino)propan-2-yl)-1<i>H</i>-indole-2-carboxamide, a New Dishevelled 1 and P-Glycoprotein Dual Inhibitor as a Anticancer AgentMichela Puxeddu, Zeyu Cui, Claudia Colla, et al.Journal of Medicinal Chemistry|July 16, 2009
New arylthioindoles and related bioisosteres at the sulfur bridging group. 4. Synthesis, tubulin polymerization, cell growth inhibition, and molecular modeling studiesGiuseppe La Regina, Taradas Sarkar, Ruoli Bai, et al.European Journal of Medicinal Chemistry|May 30, 2021
Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemiaMichela Puxeddu, Hongliang Shen, Ruoli Bai, et al.Chemmedchem|February 25, 2026
4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-GlycoproteinMichela Puxeddu, Rosa Bordone, Claudia Colla, et al.Pageof 9