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Bioorganic & Medicinal Chemistry|February 21, 2012
Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptors α/γ dual agonistsGiuseppe Fracchiolla, Antonio Laghezza, Luca Piemontese, et al.Chemmedchem|June 30, 2011
Biphenyl sulfonylamino methyl bisphosphonic acids as inhibitors of matrix metalloproteinases and bone resorptionMaria Teresa Rubino, Mariangela Agamennone, Cristina Campestre, et al.Chemmedchem|July 16, 2016
Fragment-Based Discovery of 5-Arylisatin-Based Inhibitors of Matrix Metalloproteinases 2 and 13Mariangela Agamennone, Dmitry S Belov, Antonio Laghezza, et al.European Journal of Medicinal Chemistry|December 3, 2014
Structural development studies of PPARs ligands based on tyrosine scaffoldBarbara De Filippis, Pasquale Linciano, Alessandra Ammazzalorso, et al.European Journal of Medicinal Chemistry|March 19, 2013
Molecular determinants for nuclear receptors selectivity: chemometric analysis, dockings and site-directed mutagenesis of dual peroxisome proliferator-activated receptors α/γ agonistsAntonio Carrieri, Marco Giudici, Mariagiovanna Parente, et al.Bioorganic & Medicinal Chemistry Letters|July 6, 2019
Synthesis of novel benzothiazole amides: Evaluation of PPAR activity and anti-proliferative effects in paraganglioma, pancreatic and colorectal cancer cell linesAlessandra Ammazzalorso, Laura De Lellis, Rosalba Florio, et al.European Journal of Medicinal Chemistry|December 14, 2020
Discovery of 7-aminophenanthridin-6-one as a new scaffold for matrix metalloproteinase inhibitors with multitarget neuroprotective activityDamiano Rocchi, Cristina Blázquez-Barbadillo, Mariangela Agamennone, et al.Bioorganic & Medicinal Chemistry|January 1, 2026
Targeting microbial β-CAs: bridging in silico screening with in vitro validationAnna Rita Tondo, Marialuigia Fantacuzzi, Simone Carradori, et al.Journal of Medicinal Chemistry|May 19, 2021
Thiazolidinedione "Magic Bullets" Simultaneously Targeting PPARγ and HDACs: Design, Synthesis, and Investigations of their In Vitro and In Vivo Antitumor EffectsKalpana Tilekar, Jessica D Hess, Neha Upadhyay, et al.European Journal of Medicinal Chemistry|January 12, 2017
New diphenylmethane derivatives as peroxisome proliferator-activated receptor alpha/gamma dual agonists endowed with anti-proliferative effects and mitochondrial activityLuca Piemontese, Carmen Cerchia, Antonio Laghezza, et al.Pageof 8