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European Journal of Medicinal Chemistry|October 15, 2017
Fragment-based approach to identify IDO1 inhibitor building blocksAlice Coletti, Francesca Camponeschi, Elisa Albini, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|March 26, 2026
Synthesis and structure-activity relationship study of a library of 1-substituted [1,2,4]triazolo[4,3-a]quinolines as valuable chemical probes for paraxonase-2 (PON2)Elisa Bianconi, Eros Antonio Lampitella, Fatima Nigro, et al.European Journal of Medicinal Chemistry|February 29, 2016
4,5-Diarylisoxazol-3-carboxylic acids: A new class of leukotriene biosynthesis inhibitors potentially targeting 5-lipoxygenase-activating protein (FLAP)Erden Banoglu, Erşan Çelikoğlu, Susanna Völker, et al.Journal of Medicinal Chemistry|February 18, 2014
Design, synthesis, crystallographic studies, and preliminary biological appraisal of new substituted triazolo[4,3-b]pyridazin-8-amine derivatives as tankyrase inhibitorsParide Liscio, Andrea Carotti, Stefania Asciutti, et al.Molecules (Basel, Switzerland)|December 16, 2011
Protective effects of Commiphora erythraea resin constituents against cellular oxidative damageMaria Carla Marcotullio, Federica Messina, Massimo Curini, et al.Journal of Medicinal Chemistry|December 18, 2009
Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesityRoberto Pellicciari, Antimo Gioiello, Antonio Macchiarulo, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|August 28, 2023
The hope and hype of ellagic acid and urolithins as ligands of SARS-CoV-2 Nsp5 and inhibitors of viral replicationElisa Bianconi, Anna Gidari, Maria Souma, et al.European Journal of Medicinal Chemistry|September 1, 2022
Development of 3α,7α-dihydroxy-6α-ethyl-24-nor-5β-cholan-23-sulfate sodium salt (INT-767): Process optimization, synthesis and characterization of metabolitesBruno Cerra, Francesco Venturoni, Maria Souma, et al.Bioorganic & Medicinal Chemistry|December 2, 2008
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligandsRosanna Filosa, M Carmela Fulco, Maura Marinozzi, et al.Chemmedchem|December 22, 2017
Binding Mode and Structure-Activity Relationships of ITE as an Aryl Hydrocarbon Receptor (AhR) AgonistDaniela Dolciami, Marco Gargaro, Bruno Cerra, et al.Pageof 16