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European Journal of Medicinal Chemistry|August 17, 2024
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerizationAnna Bonomini, Tommaso Felicetti, Martina Pacetti, et al.
Future Medicinal Chemistry|July 26, 2018
Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitorsGianluca Rubbini, Ana Begoña Buades-Martín, María Kimatrai-Salvador, et al.
International Journal of Molecular Sciences|April 13, 2023
Stabilization of the Dimeric State of SARS-CoV-2 Main Protease by GC376 and NirmatrelvirAlessandro Paciaroni, Valeria Libera, Francesca Ripanti, et al.
Angewandte Chemie (International Ed. in English)|June 5, 2023
Combining Solid-State NMR with Structural and Biophysical Techniques to Design Challenging Protein-Drug ConjugatesLinda Cerofolini, Kristian Vasa, Elisa Bianconi, et al.
Cancer Research|September 12, 2015
Targeting the MDM2/MDM4 interaction interface as a promising approach for p53 reactivation therapyMarsha Pellegrino, Francesca Mancini, Rossella Lucà, et al.
Chemico-Biological Interactions|March 20, 2021
Taxifolin and gastro-adhesive microparticles containing taxifolin promotes gastric healing in vivo, inhibits Helicobacter pylori in vitro and proton pump reversibly in silicoFernanda Cristina Stenger Moura, Valdir Cechinel-Filho, Francesco Antonio Greco, et al.
The Journal of Clinical Endocrinology and Metabolism|February 13, 2014
Indoleamine 2,3-dioxygenase 1 (IDO1) is up-regulated in thyroid carcinoma and drives the development of an immunosuppressant tumor microenvironmentSonia Moretti, Elisa Menicali, Pasquale Voce, et al.
Immunity|February 19, 2017
A Relay Pathway between Arginine and Tryptophan Metabolism Confers Immunosuppressive Properties on Dendritic CellsGiada Mondanelli, Roberta Bianchi, Maria Teresa Pallotta, et al.
Proceedings of the National Academy of Sciences of the United States of America|February 7, 2020
Positive allosteric modulation of indoleamine 2,3-dioxygenase 1 restrains neuroinflammationGiada Mondanelli, Alice Coletti, Francesco Antonio Greco, et al.
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