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Ariamala Gopalsamy

Showing results (11-20 of 46) with videos related to

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Organic & Biomolecular Chemistry|May 25, 2016
Cellular thermal shift and clickable chemical probe assays for the determination of drug-target engagement in live cellsHua Xu, Ariamala Gopalsamy, Erik C Hett, et al.
Bioorganic & Medicinal Chemistry Letters|February 17, 2006
Design and synthesis of 2,3,4,9-tetrahydro-1H-carbazole and 1,2,3,4-tetrahydro-cyclopenta[b]indole derivatives as non-nucleoside inhibitors of hepatitis C virus NS5B RNA-dependent RNA polymeraseAriamala Gopalsamy, Mengxiao Shi, Gregory Ciszewski, et al.
Bioorganic & Medicinal Chemistry Letters|April 14, 2009
Identification of pyrazolo[1,5-a]pyrimidine-3-carboxylates as B-Raf kinase inhibitorsAriamala Gopalsamy, Greg Ciszewski, Yongbo Hu, et al.
Journal of Medicinal Chemistry|October 19, 2007
Discovery of dibenzo[c,f][2,7]naphthyridines as potent and selective 3-phosphoinositide-dependent kinase-1 inhibitorsAriamala Gopalsamy, Mengxiao Shi, Diane H Boschelli, et al.
Bioorganic & Medicinal Chemistry Letters|July 21, 2004
Identification of [(naphthalene-1-carbonyl)-amino]-acetic acid derivatives as nonnucleoside inhibitors of HCV NS5B RNA dependent RNA polymeraseAriamala Gopalsamy, Kitae Lim, John W Ellingboe, et al.
ACS Combinatorial Science|August 6, 2016
Selectivity Determination of a Small Molecule Chemical Probe Using Protein Microarray and Affinity Capture TechniquesErik C Hett, Robert E Kyne, Ariamala Gopalsamy, et al.
Bioorganic & Medicinal Chemistry Letters|March 21, 2006
1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitorsAriamala Gopalsamy, Hui Yang, John W Ellingboe, et al.
Bioorganic & Medicinal Chemistry Letters|March 5, 2005
Pyrazolo[1,5-a]pyrimidin-7-yl phenyl amides as novel anti-proliferative agents: parallel synthesis for lead optimization of amide regionAriamala Gopalsamy, Hui Yang, John W Ellingboe, et al.
Biochemical and Biophysical Research Communications|February 7, 2008
Differing pharmacological activities of thiazolidinone analogs at the FSH receptorBrian J Arey, Stephen D Yanofsky, M Claudia Pérez, et al.
Bioorganic & Medicinal Chemistry Letters|November 4, 2009
Hit to lead optimization of pyrazolo[1,5-a]pyrimidines as B-Raf kinase inhibitorsAriamala Gopalsamy, Greg Ciszewski, Mengxiao Shi, et al.
Pageof 5

Showing results (11-20 of 46) with videos related to

Sort By:
Pageof 5
Organic & Biomolecular Chemistry|May 25, 2016
Cellular thermal shift and clickable chemical probe assays for the determination of drug-target engagement in live cellsHua Xu, Ariamala Gopalsamy, Erik C Hett, et al.
Bioorganic & Medicinal Chemistry Letters|February 17, 2006
Design and synthesis of 2,3,4,9-tetrahydro-1H-carbazole and 1,2,3,4-tetrahydro-cyclopenta[b]indole derivatives as non-nucleoside inhibitors of hepatitis C virus NS5B RNA-dependent RNA polymeraseAriamala Gopalsamy, Mengxiao Shi, Gregory Ciszewski, et al.
Bioorganic & Medicinal Chemistry Letters|April 14, 2009
Identification of pyrazolo[1,5-a]pyrimidine-3-carboxylates as B-Raf kinase inhibitorsAriamala Gopalsamy, Greg Ciszewski, Yongbo Hu, et al.
Journal of Medicinal Chemistry|October 19, 2007
Discovery of dibenzo[c,f][2,7]naphthyridines as potent and selective 3-phosphoinositide-dependent kinase-1 inhibitorsAriamala Gopalsamy, Mengxiao Shi, Diane H Boschelli, et al.
Bioorganic & Medicinal Chemistry Letters|July 21, 2004
Identification of [(naphthalene-1-carbonyl)-amino]-acetic acid derivatives as nonnucleoside inhibitors of HCV NS5B RNA dependent RNA polymeraseAriamala Gopalsamy, Kitae Lim, John W Ellingboe, et al.
ACS Combinatorial Science|August 6, 2016
Selectivity Determination of a Small Molecule Chemical Probe Using Protein Microarray and Affinity Capture TechniquesErik C Hett, Robert E Kyne, Ariamala Gopalsamy, et al.
Bioorganic & Medicinal Chemistry Letters|March 21, 2006
1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitorsAriamala Gopalsamy, Hui Yang, John W Ellingboe, et al.
Bioorganic & Medicinal Chemistry Letters|March 5, 2005
Pyrazolo[1,5-a]pyrimidin-7-yl phenyl amides as novel anti-proliferative agents: parallel synthesis for lead optimization of amide regionAriamala Gopalsamy, Hui Yang, John W Ellingboe, et al.
Biochemical and Biophysical Research Communications|February 7, 2008
Differing pharmacological activities of thiazolidinone analogs at the FSH receptorBrian J Arey, Stephen D Yanofsky, M Claudia Pérez, et al.
Bioorganic & Medicinal Chemistry Letters|November 4, 2009
Hit to lead optimization of pyrazolo[1,5-a]pyrimidines as B-Raf kinase inhibitorsAriamala Gopalsamy, Greg Ciszewski, Mengxiao Shi, et al.
Pageof 5