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Journal of Medicinal Chemistry|August 8, 2022
Iterative Optimization and Structure-Activity Relationship Studies of Oseltamivir Amino Derivatives as Potent and Selective Neuraminidase Inhibitors via Targeting 150-CavityHan Ju, Lingxin Hou, Fabao Zhao, et al.European Journal of Medicinal Chemistry|August 17, 2024
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerizationAnna Bonomini, Tommaso Felicetti, Martina Pacetti, et al.European Journal of Medicinal Chemistry|December 17, 2020
Synthesis and characterization of 1,2,4-triazolo[1,5-a]pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymeraseSerena Massari, Chiara Bertagnin, Maria Chiara Pismataro, et al.Journal of Medicinal Chemistry|October 27, 2018
Structure-Based Optimization of N-Substituted Oseltamivir Derivatives as Potent Anti-Influenza A Virus Agents with Significantly Improved Potency against Oseltamivir-Resistant N1-H274Y VariantJian Zhang, Natarajan Arul Murugan, Ye Tian, et al.Journal of Medicinal Chemistry|July 3, 2018
Optimization of N-Substituted Oseltamivir Derivatives as Potent Inhibitors of Group-1 and -2 Influenza A Neuraminidases, Including a Drug-Resistant VariantJian Zhang, Vasanthanathan Poongavanam, Dongwei Kang, et al.Nature|July 1, 2020
Suppression of a SARS-CoV-2 outbreak in the Italian municipality of Vo'Enrico Lavezzo, Elisa Franchin, Constanze Ciavarella, et al.Pageof 11