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Arnault Massink

Showing results (1-10 of 8) with videos related to

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Medicinal Research Reviews|September 10, 2019
Allosteric modulation of G protein-coupled receptors by amiloride and its derivatives. Perspectives for drug discovery?Arnault Massink, Tasia Amelia, Alex Karamychev, et al.
British Journal of Pharmacology|July 22, 2014
Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptorDong Guo, Suzanne N Venhorst, Arnault Massink, et al.
Journal of Computer-Aided Molecular Design|September 16, 2016
In search of novel ligands using a structure-based approach: a case study on the adenosine A<sub>2A</sub> receptorEelke B Lenselink, Thijs Beuming, Corine van Veen, et al.
Molecular Pharmacology|December 5, 2014
Sodium ion binding pocket mutations and adenosine A2A receptor functionArnault Massink, Hugo Gutiérrez-de-Terán, Eelke B Lenselink, et al.
European Journal of Medicinal Chemistry|July 5, 2015
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect studyRomeo Romagnoli, Pier Giovanni Baraldi, Carlota Lopez-Cara, et al.
Structure (London, England : 1993)|November 12, 2013
The role of a sodium ion binding site in the allosteric modulation of the A(2A) adenosine G protein-coupled receptorHugo Gutiérrez-de-Terán, Arnault Massink, David Rodríguez, et al.
Journal of Medicinal Chemistry|April 29, 2016
5'-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A2A ReceptorArnault Massink, Julien Louvel, Ilze Adlere, et al.
Journal of Medicinal Chemistry|September 3, 2014
Synthesis and biological evaluation of novel allosteric enhancers of the A1 adenosine receptor based on 2-amino-3-(4'-chlorobenzoyl)-4-substituted-5-arylethynyl thiopheneRomeo Romagnoli, Pier Giovanni Baraldi, Adriaan P IJzerman, et al.
Pageof 1

Showing results (1-10 of 8) with videos related to

Sort By:
Pageof 1
Medicinal Research Reviews|September 10, 2019
Allosteric modulation of G protein-coupled receptors by amiloride and its derivatives. Perspectives for drug discovery?Arnault Massink, Tasia Amelia, Alex Karamychev, et al.
British Journal of Pharmacology|July 22, 2014
Molecular mechanism of allosteric modulation at GPCRs: insight from a binding kinetics study at the human A1 adenosine receptorDong Guo, Suzanne N Venhorst, Arnault Massink, et al.
Journal of Computer-Aided Molecular Design|September 16, 2016
In search of novel ligands using a structure-based approach: a case study on the adenosine A<sub>2A</sub> receptorEelke B Lenselink, Thijs Beuming, Corine van Veen, et al.
Molecular Pharmacology|December 5, 2014
Sodium ion binding pocket mutations and adenosine A2A receptor functionArnault Massink, Hugo Gutiérrez-de-Terán, Eelke B Lenselink, et al.
European Journal of Medicinal Chemistry|July 5, 2015
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect studyRomeo Romagnoli, Pier Giovanni Baraldi, Carlota Lopez-Cara, et al.
Structure (London, England : 1993)|November 12, 2013
The role of a sodium ion binding site in the allosteric modulation of the A(2A) adenosine G protein-coupled receptorHugo Gutiérrez-de-Terán, Arnault Massink, David Rodríguez, et al.
Journal of Medicinal Chemistry|April 29, 2016
5'-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A2A ReceptorArnault Massink, Julien Louvel, Ilze Adlere, et al.
Journal of Medicinal Chemistry|September 3, 2014
Synthesis and biological evaluation of novel allosteric enhancers of the A1 adenosine receptor based on 2-amino-3-(4'-chlorobenzoyl)-4-substituted-5-arylethynyl thiopheneRomeo Romagnoli, Pier Giovanni Baraldi, Adriaan P IJzerman, et al.
Pageof 1