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Bioorganic & Medicinal Chemistry Letters
|
August 25, 2009
Synthesis and SAR of 1,4,5,6-tetrahydropyridazines as potent cannabinoid CB1 receptor antagonists
Jos H M Lange, Arnold P den Hartog, Martina A W van der Neut, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 20, 2017
Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P<sub>5</sub> receptor agonist chemotype
Axel R Stoit, Jos H M Lange, Hein K A C Coolen, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 9, 2010
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB(1) receptor antagonists
Jos H M Lange, Martina A W van der Neut, Arnold P den Hartog, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 17, 2007
7-Azaindole derivatives as potential partial nicotinic agonists
Axel R Stoit, Arnold P den Hartog, Harry Mons, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 25, 2009
Synthesis and SAR of novel imidazoles as potent and selective cannabinoid CB2 receptor antagonists with high binding efficiencies
Jos H M Lange, Martina A W van der Neut, Henri C Wals, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 16, 2016
Optimization of N'-(arylsulfonyl)pyrazoline-1-carboxamidines by exploiting a novel interaction site in the 5-HT6 antagonistic binding pocket
Arnold van Loevezijn, Jennifer Venhorst, Wouter I Iwema Bakker, et al.
Journal of Medicinal Chemistry
|
October 28, 2005
Synthesis, structure-activity relationships, and biological properties of 1-heteroaryl-4-[omega-(1H-indol-3-yl)alkyl]piperazines, novel potential antipsychotics combining potent dopamine D2 receptor antagonism with potent serotonin reuptake inhibition
Pieter Smid, Hein K A C Coolen, Hiskias G Keizer, et al.
Journal of Medicinal Chemistry
|
January 23, 2004
Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists
Jos H M Lange, Hein K A C Coolen, Herman H van Stuivenberg, et al.
Page
of 1
Search research articles
Search
Showing results (1-10 of 8) with videos related to
Sort By:
Page
of 1
Bioorganic & Medicinal Chemistry Letters
|
August 25, 2009
Synthesis and SAR of 1,4,5,6-tetrahydropyridazines as potent cannabinoid CB1 receptor antagonists
Jos H M Lange, Arnold P den Hartog, Martina A W van der Neut, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 20, 2017
Spiro-1-benzofuranpiperidinylalkanoic acids as a novel and selective sphingosine S1P<sub>5</sub> receptor agonist chemotype
Axel R Stoit, Jos H M Lange, Hein K A C Coolen, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 9, 2010
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB(1) receptor antagonists
Jos H M Lange, Martina A W van der Neut, Arnold P den Hartog, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 17, 2007
7-Azaindole derivatives as potential partial nicotinic agonists
Axel R Stoit, Arnold P den Hartog, Harry Mons, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 25, 2009
Synthesis and SAR of novel imidazoles as potent and selective cannabinoid CB2 receptor antagonists with high binding efficiencies
Jos H M Lange, Martina A W van der Neut, Henri C Wals, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 16, 2016
Optimization of N'-(arylsulfonyl)pyrazoline-1-carboxamidines by exploiting a novel interaction site in the 5-HT6 antagonistic binding pocket
Arnold van Loevezijn, Jennifer Venhorst, Wouter I Iwema Bakker, et al.
Journal of Medicinal Chemistry
|
October 28, 2005
Synthesis, structure-activity relationships, and biological properties of 1-heteroaryl-4-[omega-(1H-indol-3-yl)alkyl]piperazines, novel potential antipsychotics combining potent dopamine D2 receptor antagonism with potent serotonin reuptake inhibition
Pieter Smid, Hein K A C Coolen, Hiskias G Keizer, et al.
Journal of Medicinal Chemistry
|
January 23, 2004
Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists
Jos H M Lange, Hein K A C Coolen, Herman H van Stuivenberg, et al.
Page
of 1