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Arthur Christopoulos

Showing results (181-190 of 331) with videos related to

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European Journal of Medicinal Chemistry|June 22, 2007
Synthesis and cannabinoid activity of 1-substituted-indole-3-oxadiazole derivatives: novel agonists for the CB1 receptorGerard P Moloney, James A Angus, Alan D Robertson, et al.
Journal of Medicinal Chemistry|February 10, 2012
Synthesis and characterization of novel 2-amino-3-benzoylthiophene derivatives as biased allosteric agonists and modulators of the adenosine A(1) receptorCeline Valant, Luigi Aurelio, Shane M Devine, et al.
Plos One|March 20, 2014
Prolonged calcitonin receptor signaling by salmon, but not human calcitonin, reveals ligand biasKim Vietz Andreassen, Sara Toftegaard Hjuler, Sebastian G Furness, et al.
Molecular Pharmacology|October 7, 2005
Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonistChristopher J Langmead, Victoria A H Fry, Ian T Forbes, et al.
Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology|November 27, 2009
Molecular mechanisms of action and in vivo validation of an M4 muscarinic acetylcholine receptor allosteric modulator with potential antipsychotic propertiesKatie Leach, Richard E Loiacono, Christian C Felder, et al.
The Journal of Biological Chemistry|December 29, 2010
Allosteric modulation of the calcium-sensing receptor by gamma-glutamyl peptides: inhibition of PTH secretion, suppression of intracellular cAMP levels, and a common mechanism of action with L-amino acidsGeoffrey K Broadhead, Hee-chang Mun, Vimesh A Avlani, et al.
The Journal of Biological Chemistry|October 19, 2014
Mechanistic insights into allosteric structure-function relationships at the M1 muscarinic acetylcholine receptorAlaa Abdul-Ridha, J Robert Lane, Shailesh N Mistry, et al.
Molecular Pharmacology|August 6, 2015
Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor AntagonistsDarren M Riddy, Celine Valant, Patricia Rueda, et al.
The Journal of Pharmacology and Experimental Therapeutics|July 31, 2009
Determination of adenosine A1 receptor agonist and antagonist pharmacology using Saccharomyces cerevisiae: implications for ligand screening and functional selectivityGregory D Stewart, Celine Valant, Simon J Dowell, et al.
Biochemical Society Transactions|January 30, 2013
Recent advances in understanding GLP-1R (glucagon-like peptide-1 receptor) functionCassandra Koole, Kavita Pabreja, Emilia E Savage, et al.
Pageof 34

Showing results (181-190 of 331) with videos related to

Sort By:
Pageof 34
European Journal of Medicinal Chemistry|June 22, 2007
Synthesis and cannabinoid activity of 1-substituted-indole-3-oxadiazole derivatives: novel agonists for the CB1 receptorGerard P Moloney, James A Angus, Alan D Robertson, et al.
Journal of Medicinal Chemistry|February 10, 2012
Synthesis and characterization of novel 2-amino-3-benzoylthiophene derivatives as biased allosteric agonists and modulators of the adenosine A(1) receptorCeline Valant, Luigi Aurelio, Shane M Devine, et al.
Plos One|March 20, 2014
Prolonged calcitonin receptor signaling by salmon, but not human calcitonin, reveals ligand biasKim Vietz Andreassen, Sara Toftegaard Hjuler, Sebastian G Furness, et al.
Molecular Pharmacology|October 7, 2005
Probing the molecular mechanism of interaction between 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine (AC-42) and the muscarinic M(1) receptor: direct pharmacological evidence that AC-42 is an allosteric agonistChristopher J Langmead, Victoria A H Fry, Ian T Forbes, et al.
Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology|November 27, 2009
Molecular mechanisms of action and in vivo validation of an M4 muscarinic acetylcholine receptor allosteric modulator with potential antipsychotic propertiesKatie Leach, Richard E Loiacono, Christian C Felder, et al.
The Journal of Biological Chemistry|December 29, 2010
Allosteric modulation of the calcium-sensing receptor by gamma-glutamyl peptides: inhibition of PTH secretion, suppression of intracellular cAMP levels, and a common mechanism of action with L-amino acidsGeoffrey K Broadhead, Hee-chang Mun, Vimesh A Avlani, et al.
The Journal of Biological Chemistry|October 19, 2014
Mechanistic insights into allosteric structure-function relationships at the M1 muscarinic acetylcholine receptorAlaa Abdul-Ridha, J Robert Lane, Shailesh N Mistry, et al.
Molecular Pharmacology|August 6, 2015
Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor AntagonistsDarren M Riddy, Celine Valant, Patricia Rueda, et al.
The Journal of Pharmacology and Experimental Therapeutics|July 31, 2009
Determination of adenosine A1 receptor agonist and antagonist pharmacology using Saccharomyces cerevisiae: implications for ligand screening and functional selectivityGregory D Stewart, Celine Valant, Simon J Dowell, et al.
Biochemical Society Transactions|January 30, 2013
Recent advances in understanding GLP-1R (glucagon-like peptide-1 receptor) functionCassandra Koole, Kavita Pabreja, Emilia E Savage, et al.
Pageof 34