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Bioorganic & Medicinal Chemistry Letters|April 3, 2007
Preparation of novel anthranilic acids as antibacterial agents: extensive evaluation of structural and physical properties on antibacterial activity and human serum albumin affinityAtli Thorarensen, Jianke Li, Brian D Wakefield, et al.Bioorganic & Medicinal Chemistry|December 7, 2020
The advantages of describing covalent inhibitor in vitro potencies by IC50 at a fixed time point. IC50 determination of covalent inhibitors provides meaningful data to medicinal chemistry for SAR optimizationAtli Thorarensen, Paul Balbo, Mary E Banker, et al.Bioorganic & Medicinal Chemistry Letters|September 22, 2009
Structure based design of novel irreversible FAAH inhibitorsJane L Wang, Scott J Bowen, Barbara A Schweitzer, et al.Bioorganic & Medicinal Chemistry Letters|March 21, 2007
Preparation of novel anthranilic acids as antibacterial agents. Extensive evaluation of alternative amide bioisosteres connecting the A- and the B-ringsAtli Thorarensen, Brian D Wakefield, Donna L Romero, et al.Drug Metabolism and Disposition: the Biological Fate of Chemicals|October 28, 2016
Clearance Prediction of Targeted Covalent Inhibitors by In Vitro-In Vivo Extrapolation of Hepatic and Extrahepatic Clearance MechanismsLouis Leung, Xin Yang, Timothy J Strelevitz, et al.Bioorganic & Medicinal Chemistry Letters|March 14, 2007
Preparation of novel antibacterial agents. Replacement of the central aromatic ring with heterocyclesJianke Li, Brian D Wakefield, J Craig Ruble, et al.Bioorganic & Medicinal Chemistry Letters|October 28, 2008
Bacterial translation inhibitors, 1-acylindazol-3-ols as anthranilic acid mimicsCory Stiff, David R Graber, Atli Thorarensen, et al.Chemical Biology & Drug Design|July 5, 2012
Identification of type-II inhibitors using kinase structuresFrank Lovering, Joseph McDonald, Gavin A Whitlock, et al.Bioconjugate Chemistry|March 18, 2004
Immobilization of a novel antibacterial agent on solid phase and subsequent isolation of EF-TuMartin R Deibel, Alice L Bodnar, Anthony W Yem, et al.Chemmedchem|September 19, 2015
Imidazotriazines: Spleen Tyrosine Kinase (Syk) Inhibitors Identified by Free-Energy Perturbation (FEP)Frank Lovering, Cristina Aevazelis, Jeanne Chang, et al.Pageof 4