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Bioorganic & Medicinal Chemistry|December 21, 2017
Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivativesMitsunori Kono, Tsuneo Oda, Michiko Tawada, et al.Chemmedchem|October 30, 2019
Design and Synthesis of Conformationally Constrained RORγt Inverse AgonistsAyumu Sato, Yoshiyuki Fukase, Mitsunori Kono, et al.Bioorganic & Medicinal Chemistry|December 22, 2017
Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffoldsJunya Shirai, Yoshihide Tomata, Mitsunori Kono, et al.Journal of Medicinal Chemistry|August 26, 2021
Discovery and Structure-Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious AntimalarialsBenoît Laleu, Yuichiro Akao, Atsuko Ochida, et al.Antimicrobial Agents and Chemotherapy|February 13, 2019
Optimization of Methionyl tRNA-Synthetase Inhibitors for Treatment of Cryptosporidium InfectionFrederick S Buckner, Ranae M Ranade, J Robert Gillespie, et al.Journal of Medicinal Chemistry|March 7, 2018
Discovery of [ cis-3-({(5 R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro-1 H-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5 H)-yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor γt Inverse AgonistMitsunori Kono, Atsuko Ochida, Tsuneo Oda, et al.Ebiomedicine|March 23, 2024
High-throughput screening of small-molecules libraries identified antibacterials against clinically relevant multidrug-resistant A. baumannii and K. pneumoniaeBenjamin Blasco, Soojin Jang, Hiroki Terauchi, et al.Journal of Medicinal Chemistry|January 6, 2023
Collaborative Virtual Screening Identifies a 2-Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi InfectionTaisuke Tawaraishi, Atsuko Ochida, Yuichiro Akao, et al.ACS Infectious Diseases|April 30, 2021
Repositioning and Characterization of 1-(Pyridin-4-yl)pyrrolidin-2-one Derivatives as Plasmodium Cytoplasmic Prolyl-tRNA Synthetase InhibitorsMasanori Okaniwa, Akira Shibata, Atsuko Ochida, et al.Pageof 2