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Bioorganic & Medicinal Chemistry|January 23, 2024
Pentafluorosulfanyl-substituted biaryl derivatives as MATE-type transporter inhibitors targeting drug-resistant bacteriaSusumu Shinya, Kentaro Kawai, Naoki Kobayashi, et al.
Organic Letters|April 5, 2014
Ligand-promoted asymmetric imino-Reformatsky reaction of ethyl dibromofluoroacetateAtsushi Tarui, Haruka Nishimura, Takeshi Ikebata, et al.
Beilstein Journal of Organic Chemistry|March 23, 2018
Development of a fluorogenic small substrate for dipeptidyl peptidase-4Futa Ogawa, Masanori Takeda, Kanae Miyanaga, et al.
Beilstein Journal of Organic Chemistry|June 18, 2024
Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitorKazuyuki Sato, Satoki Teranishi, Atsushi Sakaue, et al.
Molecular Informatics|March 19, 2021
Effect of Learning Dataset for Identification of Active Molecules: A Case Study of Integrin αIIbβ3 InhibitorsKentaro Kawai, Mami Tomonou, Yume Machida, et al.
Chemical & Pharmaceutical Bulletin|November 6, 2007
Formation of quaternary carbon center with a trifluoromethyl group using a Pd-catalyzed allylation reactionKazuyuki Sato, Yu Takiguchi, Yosuke Yoshizawa, et al.
Bioorganic & Medicinal Chemistry Letters|October 21, 2025
Discovery of a novel pharmacokinetic booster: A small intestine-selective CYP3A4 inhibitor with dibenzyl ether structureShoki Hoshikawa, Koki Kimura, Chisaki Hanada, et al.
Bioorganic & Medicinal Chemistry Letters|June 28, 2022
Discovery of benzyloxyphenyl- and phenethylphenyl-imidazole derivatives as a new class of ante-drug type boostersKentaro Kawai, Jun Okada, Mizuki Nakae, et al.
Bioorganic & Medicinal Chemistry|March 23, 2019
Structural modification of indomethacin toward selective inhibition of COX-2 with a significant increase in van der Waals contributionsAkari Ikeda, Eishi Funakoshi, Mitsugu Araki, et al.
Beilstein Journal of Organic Chemistry|December 19, 2022
Rhodium-catalyzed intramolecular reductive aldol-type cyclization: Application for the synthesis of a chiral necic acid lactoneMotoyuki Isoda, Kazuyuki Sato, Kenta Kameda, et al.
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