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September 28, 2001
Pumping it up
B Luscombe
British Journal of Pharmacology
|
December 27, 2023
Biased agonists of GPR84 and insights into biological control
Vincent B Luscombe, Pinqi Wang, Angela J Russell, et al.
DNA and Cell Biology
|
October 1, 2020
20 Years an Orphan: Is GPR84 a Plausible Medium-Chain Fatty Acid-Sensing Receptor?
Vincent B Luscombe, Daniel Lucy, Carole J R Bataille, et al.
European Journal of Pharmacology
|
August 5, 2023
Kinetic insights into agonist-dependent signalling bias at the pro-inflammatory G-protein coupled receptor GPR84
Vincent B Luscombe, Luis Alberto Baena-López, Carole J R Bataille, et al.
Journal of Medicinal Chemistry
|
December 26, 2023
Development of Highly Potent, G-Protein Pathway Biased, Selective, and Orally Bioavailable GPR84 Agonists
Pinqi Wang, Arun Raja, Vincent B Luscombe, et al.
ACS Chemical Neuroscience
|
May 28, 2019
Identification of Novel Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5 Acting at Site Distinct from 2-Methyl-6-(phenylethynyl)-pyridine Binding
Mariusz Butkiewicz, Alice L Rodriguez, Shane E Rainey, et al.
ACS Omega
|
August 29, 2019
Evaluation of Synthetic Cytochrome P<sub>450</sub>-Mimetic Metalloporphyrins To Facilitate "Biomimetic" Biotransformation of a Series of mGlu<sub>5</sub> Allosteric Ligands
Christopher C Presley, Charles K Perry, Elizabeth S Childress, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 22, 2017
Synthesis and evaluation of 4,6-disubstituted pyrimidines as CNS penetrant pan-muscarinic antagonists with a novel chemotype
Aaron M Bender, Rebecca L Weiner, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 12, 2021
Discovery of a novel class of heteroaryl-pyrrolidinones as positive allosteric modulators of the muscarinic acetylcholine receptor M<sub>1</sub>
Paul K Spearing, Hyekyung P Cho, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2019
Discovery of structurally distinct tricyclic M<sub>4</sub> positive allosteric modulator (PAM) chemotypes
Kayla J Temple, Madeline F Long, Julie L Engers, et al.
Page
of 4
Search research articles
Search
Showing results (1-10 of 36) with videos related to
Sort By:
Page
of 4
Time
|
September 28, 2001
Pumping it up
B Luscombe
British Journal of Pharmacology
|
December 27, 2023
Biased agonists of GPR84 and insights into biological control
Vincent B Luscombe, Pinqi Wang, Angela J Russell, et al.
DNA and Cell Biology
|
October 1, 2020
20 Years an Orphan: Is GPR84 a Plausible Medium-Chain Fatty Acid-Sensing Receptor?
Vincent B Luscombe, Daniel Lucy, Carole J R Bataille, et al.
European Journal of Pharmacology
|
August 5, 2023
Kinetic insights into agonist-dependent signalling bias at the pro-inflammatory G-protein coupled receptor GPR84
Vincent B Luscombe, Luis Alberto Baena-López, Carole J R Bataille, et al.
Journal of Medicinal Chemistry
|
December 26, 2023
Development of Highly Potent, G-Protein Pathway Biased, Selective, and Orally Bioavailable GPR84 Agonists
Pinqi Wang, Arun Raja, Vincent B Luscombe, et al.
ACS Chemical Neuroscience
|
May 28, 2019
Identification of Novel Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5 Acting at Site Distinct from 2-Methyl-6-(phenylethynyl)-pyridine Binding
Mariusz Butkiewicz, Alice L Rodriguez, Shane E Rainey, et al.
ACS Omega
|
August 29, 2019
Evaluation of Synthetic Cytochrome P<sub>450</sub>-Mimetic Metalloporphyrins To Facilitate "Biomimetic" Biotransformation of a Series of mGlu<sub>5</sub> Allosteric Ligands
Christopher C Presley, Charles K Perry, Elizabeth S Childress, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 22, 2017
Synthesis and evaluation of 4,6-disubstituted pyrimidines as CNS penetrant pan-muscarinic antagonists with a novel chemotype
Aaron M Bender, Rebecca L Weiner, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 12, 2021
Discovery of a novel class of heteroaryl-pyrrolidinones as positive allosteric modulators of the muscarinic acetylcholine receptor M<sub>1</sub>
Paul K Spearing, Hyekyung P Cho, Vincent B Luscombe, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2019
Discovery of structurally distinct tricyclic M<sub>4</sub> positive allosteric modulator (PAM) chemotypes
Kayla J Temple, Madeline F Long, Julie L Engers, et al.
Page
of 4