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Bioorganic & Medicinal Chemistry
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September 24, 2025
Decades old glitazones still find niche in drug discoveries as PPAR-γ agonists: medicinal chemistry perspective, structure-activity relationships and therapeutic implications
P Archana, T Durai Ananda Kumar, N Vijaya Ganesh, et al.
Frontiers in Bioinformatics
|
June 17, 2026
Integrated computational-based design of putative dual TrkA/TrkB agonists for Alzheimer's disease: pharmacophore modelling, docking, MM/GBSA, DFT and dynamics studies
A Vignesh Pandi, Vishnu Malakar, Jeyaram Bharathi Jeyabalan, et al.
Chemical Biology & Drug Design
|
January 3, 2026
Computational Based Identified EAAT2 Transporter Activator Attenuates Amyloid-β Induced Excitotoxicity in Primary Neuronal-Astroglial Mixed Culture by Ameliorating Glutamate Clearance
Chennu Manisha, Anusa Ganguly, Nagarjuna Palathoti, et al.
Molecules (Basel, Switzerland)
|
May 13, 2023
Novel Derivatives of Eugenol as a New Class of PPARγ Agonists in Treating Inflammation: Design, Synthesis, SAR Analysis and In Vitro Anti-Inflammatory Activity
Noor Fathima Anjum, Dhivya Shanmugarajan, B R Prashantha Kumar, et al.
RSC Advances
|
June 27, 2022
Novel derivatives of eugenol as potent anti-inflammatory agents <i>via</i> PPARγ agonism: rational design, synthesis, analysis, PPARγ protein binding assay and computational studies
Noor Fathima Anjum, Dhivya Shanmugarajan, Vasanth Kumar Shivaraju, et al.
Current Topics in Medicinal Chemistry
|
January 4, 2025
Updates on Intrinsic Medicinal Chemistry of 1,4-dihydropyridines, Perspectives on Synthesis and Pharmacokinetics of Novel 1,4-dihydropyrimidines as Calcium Channel Blockers: Clinical Pharmacology
Chiriki Devi Sri, Narasimha Murthy Beeraka, Hemanth Vikram P R, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 14, 2026
Multifunctional quinoline-based hydrazones as promising antidiabetic agents: experimental and computational insights
Aditi Kalakwade, Rohini S Kavalapure, Shankar Gharge, et al.
Bioorganic Chemistry
|
November 9, 2021
Design, parallel synthesis of Biginelli 1,4-dihydropyrimidines using PTSA as a catalyst, evaluation of anticancer activity and structure activity relationships via 3D QSAR studies
Syed Faizan, B R Prashantha Kumar, Namburu Lalitha Naishima, et al.
Antibiotics (Basel, Switzerland)
|
July 29, 2023
Discovery of Novel Myristic Acid Derivatives as N-Myristoyltransferase Inhibitors: Design, Synthesis, Analysis, Computational Studies and Antifungal Activity
Saleem Javid, Hissana Ather, Umme Hani, et al.
Frontiers in Neuroscience
|
October 26, 2020
Two Rationally Identified Novel Glitazones Reversed the Behavioral Dysfunctions and Exhibited Neuroprotection Through Ameliorating Brain Cytokines and Oxy-Radicals in ICV-LPS Neuroinflammatory Rat Model
Antony Justin, Premkumar Ashwini, Jincy A Jose, et al.
Page
of 5
Search research articles
Search
Showing results (31-40 of 47) with videos related to
Sort By:
Page
of 5
Bioorganic & Medicinal Chemistry
|
September 24, 2025
Decades old glitazones still find niche in drug discoveries as PPAR-γ agonists: medicinal chemistry perspective, structure-activity relationships and therapeutic implications
P Archana, T Durai Ananda Kumar, N Vijaya Ganesh, et al.
Frontiers in Bioinformatics
|
June 17, 2026
Integrated computational-based design of putative dual TrkA/TrkB agonists for Alzheimer's disease: pharmacophore modelling, docking, MM/GBSA, DFT and dynamics studies
A Vignesh Pandi, Vishnu Malakar, Jeyaram Bharathi Jeyabalan, et al.
Chemical Biology & Drug Design
|
January 3, 2026
Computational Based Identified EAAT2 Transporter Activator Attenuates Amyloid-β Induced Excitotoxicity in Primary Neuronal-Astroglial Mixed Culture by Ameliorating Glutamate Clearance
Chennu Manisha, Anusa Ganguly, Nagarjuna Palathoti, et al.
Molecules (Basel, Switzerland)
|
May 13, 2023
Novel Derivatives of Eugenol as a New Class of PPARγ Agonists in Treating Inflammation: Design, Synthesis, SAR Analysis and In Vitro Anti-Inflammatory Activity
Noor Fathima Anjum, Dhivya Shanmugarajan, B R Prashantha Kumar, et al.
RSC Advances
|
June 27, 2022
Novel derivatives of eugenol as potent anti-inflammatory agents <i>via</i> PPARγ agonism: rational design, synthesis, analysis, PPARγ protein binding assay and computational studies
Noor Fathima Anjum, Dhivya Shanmugarajan, Vasanth Kumar Shivaraju, et al.
Current Topics in Medicinal Chemistry
|
January 4, 2025
Updates on Intrinsic Medicinal Chemistry of 1,4-dihydropyridines, Perspectives on Synthesis and Pharmacokinetics of Novel 1,4-dihydropyrimidines as Calcium Channel Blockers: Clinical Pharmacology
Chiriki Devi Sri, Narasimha Murthy Beeraka, Hemanth Vikram P R, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 14, 2026
Multifunctional quinoline-based hydrazones as promising antidiabetic agents: experimental and computational insights
Aditi Kalakwade, Rohini S Kavalapure, Shankar Gharge, et al.
Bioorganic Chemistry
|
November 9, 2021
Design, parallel synthesis of Biginelli 1,4-dihydropyrimidines using PTSA as a catalyst, evaluation of anticancer activity and structure activity relationships via 3D QSAR studies
Syed Faizan, B R Prashantha Kumar, Namburu Lalitha Naishima, et al.
Antibiotics (Basel, Switzerland)
|
July 29, 2023
Discovery of Novel Myristic Acid Derivatives as N-Myristoyltransferase Inhibitors: Design, Synthesis, Analysis, Computational Studies and Antifungal Activity
Saleem Javid, Hissana Ather, Umme Hani, et al.
Frontiers in Neuroscience
|
October 26, 2020
Two Rationally Identified Novel Glitazones Reversed the Behavioral Dysfunctions and Exhibited Neuroprotection Through Ameliorating Brain Cytokines and Oxy-Radicals in ICV-LPS Neuroinflammatory Rat Model
Antony Justin, Premkumar Ashwini, Jincy A Jose, et al.
Page
of 5