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Expert Opinion on Therapeutic Patents|October 5, 2022
An updated patent review of rearranged during transfection (RET) kinase inhibitors (2016-present)Baku Acharya, Brendan FrettRSC Medicinal Chemistry|August 4, 2022
FLT3 inhibitors for acute myeloid leukemia: successes, defeats, and emerging paradigmsBaku Acharya, Debasmita Saha, Daniel Armstrong, et al.Genes|July 27, 2022
Targeting a Novel G-Quadruplex in the CARD11 Oncogene Promoter with Naptho(2,1-b)furan-1-ethanol,2-nitro- Requires the Nitro GroupKennith Swafford, Baku Acharya, Ying-Zhi Xu, et al.Journal of Medicinal Chemistry|August 17, 2021
Targeting Rearranged during Transfection in Cancer: A Perspective on Small-Molecule Inhibitors and Their Clinical DevelopmentDebasmita Saha, Katie Rose Ryan, Naga Rajiv Lakkaniga, et al.The Journal of Pharmacology and Experimental Therapeutics|July 24, 2025
Transforming growth factor β receptor 1 and mitogen-activated protein 4 kinase 4 dual inhibitor, TK-850, reduces renal fibrosis in unilateral ureteral-obstructed miceHenry A Palfrey, Samaneh Goorani, Abhishek Mishra, et al.Bioorganic & Medicinal Chemistry|May 14, 2024
Discovery of 9H-pyrimido[4,5-b]indole derivatives as dual RET/TRKA inhibitorsBaku Acharya, Debasmita Saha, Noemi Garcia Garcia, et al.RSC Medicinal Chemistry|February 23, 2024
Kinase inhibitor macrocycles: a perspective on limiting conformational flexibility when targeting the kinome with small moleculesBaku Acharya, Debasmita Saha, Daniel Armstrong, et al.Scientific Reports|August 28, 2024
Discovery of the DNA-PKcs inhibitor DA-143 which exhibits enhanced solubility relative to NU7441Zachary J Waldrip, Baku Acharya, Daniel Armstrong, et al.Expert Opinion on Therapeutic Patents|June 12, 2025
An updated patent review of rearranged during transfection (RET) kinase inhibitors (2022-present)Daniel Armstrong, Maha Hanafi, Brendan FrettOrganic Letters|May 24, 2014
Efficient access to 2,3-diarylimidazo[1,2-a]pyridines via a one-pot, ligand-free, palladium-catalyzed three-component reaction under microwave irradiationYuanxiang Wang, Brendan Frett, Hong-yu LiPageof 7