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BMC Cancer|January 18, 2019
Estrogen receptor signaling regulates the expression of the breast tumor kinase in breast cancer cellsSayem Miah, Edward Bagu, Raghuveera Goel, et al.
Angewandte Chemie (International Ed. in English)|July 2, 2015
Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent PolypharmacologyBrendan Frett, Francesca Carlomagno, Maria Luisa Moccia, et al.
European Journal of Medicinal Chemistry|September 3, 2021
Discovery of imidazo[1,2-a]pyridine-thiophene derivatives as FLT3 and FLT3 mutants inhibitors for acute myeloid leukemia through structure-based optimization of an NEK2 inhibitorLingtian Zhang, Naga Rajiv Lakkaniga, Jaideep B Bharate, et al.
Molecular & Cellular Proteomics : MCP|March 31, 2018
A Structured Workflow for Mapping Human Sin3 Histone Deacetylase Complex Interactions Using Halo-MudPIT Affinity-Purification Mass SpectrometryCharles A S Banks, Janet L Thornton, Cassandra G Eubanks, et al.
Chemical Communications (Cambridge, England)|February 8, 2020
Correction: One-pot construction of functionalized aziridines and maleimides via a novel pseudo-Knoevenagel cascade reactionJie Lei, Gui-Ting Song, Liu-Jun He, et al.
Chemical Communications (Cambridge, England)|January 24, 2020
One-pot construction of functionalized aziridines and maleimides via a novel pseudo-Knoevenagel cascade reactionJie Lei, Gui-Ting Song, Liu-Jun He, et al.
Scientific Reports|August 10, 2021
Targeted activity of the small molecule kinase inhibitor Pz-1 towards RET and TRK kinasesMarialuisa Moccia, Donglin Yang, Naga Rajiv Lakkaniga, et al.
Oncotarget|January 20, 2018
FRK inhibits breast cancer cell migration and invasion by suppressing epithelial-mesenchymal transitionYetunde Ogunbolude, Chenlu Dai, Edward T Bagu, et al.
Bioorganic & Medicinal Chemistry|June 21, 2018
Facile construction of fused benzimidazole-isoquinolinones that induce cell-cycle arrest and apoptosis in colorectal cancer cellsLiu-Jun He, Dong-Lin Yang, Shi-Qiang Li, et al.
Journal of Medicinal Chemistry|April 17, 2020
Bioisosteric Discovery of NPA101.3, a Second-Generation RET/VEGFR2 Inhibitor Optimized for Single-Agent PolypharmacologyMarialuisa Moccia, Brendan Frett, Lingtian Zhang, et al.
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