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Journal of Medicinal Chemistry|March 24, 2010
The significance of 2-furyl ring substitution with a 2-(para-substituted) aryl group in a new series of pyrazolo-triazolo-pyrimidines as potent and highly selective hA(3) adenosine receptors antagonists: new insights into structure-affinity relationship and receptor-antagonist recognitionSiew Lee Cheong, Anna Dolzhenko, Sonja Kachler, et al.Pharmaceuticals (Basel, Switzerland)|November 16, 2019
Chemical Probes for the Adenosine ReceptorsStephanie Federico, Lucia Lassiani, Giampiero SpallutoBioorganic & Medicinal Chemistry|June 9, 2009
Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sitesLisa Michielan, Chiara Bolcato, Stephanie Federico, et al.Bioorganic & Medicinal Chemistry|March 23, 2010
Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand-receptor recognition processGiorgia Pastorin, Stephanie Federico, Silvia Paoletta, et al.Bioorganic & Medicinal Chemistry|May 26, 2009
6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptorsPamela Crepaldi, Barbara Cacciari, Maria-Cruz Bonache, et al.Journal of Chemical Information and Modeling|May 28, 2013
Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonistsMagdalena Bacilieri, Antonella Ciancetta, Silvia Paoletta, et al.Trends in Pharmacological Sciences|January 5, 2005
Techniques: Recent developments in computer-aided engineering of GPCR ligands using the human adenosine A3 receptor as an exampleStefano Moro, Giampiero Spalluto, Kenneth A JacobsonJournal of Medicinal Chemistry|August 9, 2002
Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonistAnna Maconi, Giorgia Pastorin, Tatiana Da Ros, et al.Journal of Medicinal Chemistry|January 11, 2011
Synthesis and biological evaluation of a new series of 1,2,4-triazolo[1,5-a]-1,3,5-triazines as human A(2A) adenosine receptor antagonists with improved water solubilityStephanie Federico, Silvia Paoletta, Siew Lee Cheong, et al.Current Pharmaceutical Design|June 27, 2006
Ligand-based homology modeling as attractive tool to inspect GPCR structural plasticityStefano Moro, Francesca Deflorian, Magdalena Bacilieri, et al.Pageof 10