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ACS Medicinal Chemistry Letters|June 24, 2015
Selective Acetamidine-Based Nitric Oxide Synthase Inhibitors: Synthesis, Docking, and Biological StudiesCristina Maccallini, Monica Montagnani, Roberto Paciotti, et al.Archiv Der Pharmazie|May 28, 2024
Synthesis and in vitro cytotoxicity of benzoxazole-based PPARα/γ antagonists in colorectal cancer cell linesNazaret Moreno-Rodríguez, Antonio Laghezza, Carmen Cerchia, et al.European Journal of Medicinal Chemistry|March 15, 2016
Synthesis, in vitro evaluation, and molecular modeling investigation of benzenesulfonimide peroxisome proliferator-activated receptors α antagonistsAlessandra Ammazzalorso, Antonio Carrieri, Fabio Verginelli, et al.Journal of Medicinal Chemistry|February 11, 2009
Synthesis, biological evaluation, and docking studies of N-substituted acetamidines as selective inhibitors of inducible nitric oxide synthaseCristina Maccallini, Antonia Patruno, Neva Besker, et al.ACS Medicinal Chemistry Letters|June 19, 2024
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase InhibitorsJaydeo T Kilbile, Suryakant B Sapkal, Gioele Renzi, et al.ACS Medicinal Chemistry Letters|May 22, 2020
Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking StudiesAlessandra Ammazzalorso, Isabella Bruno, Rosalba Florio, et al.Pharmaceuticals (Basel, Switzerland)|March 29, 2023
Anti-Inflammatory, Antioxidant, and WAT/BAT-Conversion Stimulation Induced by Novel PPAR Ligands: Results from Ex Vivo and In Vitro StudiesLucia Recinella, Barbara De Filippis, Maria Loreta Libero, et al.ACS Pharmacology & Translational Science|May 14, 2026
Synthesis, Biological Evaluation, and Computational Study of Pyridine- and Indazole-Based Inhibitors of the Inducible Nitric Oxide Synthase as Promising Antipsoriatic AgentsPasquale Amoia, Marialucia Gallorini, Claudia Scarponi, et al.Pharmaceuticals (Basel, Switzerland)|August 29, 2024
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational StudiesLetizia Giampietro, Beatrice Marinacci, Alice Della Valle, et al.European Journal of Medicinal Chemistry|April 25, 2018
Discovery of N-{3-[(ethanimidoylamino)methyl]benzyl}-l-prolinamide dihydrochloride: A new potent and selective inhibitor of the inducible nitric oxide synthase as a promising agent for the therapy of malignant gliomaCristina Maccallini, Mauro Di Matteo, Marialucia Gallorini, et al.Pageof 9