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Bioorganic & Medicinal Chemistry Letters
|
December 22, 2019
Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors
Benjamin N Atkinson, David Steadman, William Mahy, et al.
Journal of Medicinal Chemistry
|
August 14, 2020
Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity
William Mahy, Mikesh Patel, David Steadman, et al.
ACS Chemical Neuroscience
|
June 22, 2022
Structural Analysis and Development of Notum Fragment Screening Hits
Yuguang Zhao, William Mahy, Nicky J Willis, et al.
Journal of Medicinal Chemistry
|
May 10, 2022
Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit
Nicky J Willis, William Mahy, James Sipthorp, et al.
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Search research articles
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Showing results (11-20 of 14) with videos related to
Sort By:
Page
of 2
You have reached the last page of results.
This site can display upto 14 results.
Bioorganic & Medicinal Chemistry Letters
|
December 22, 2019
Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors
Benjamin N Atkinson, David Steadman, William Mahy, et al.
Journal of Medicinal Chemistry
|
August 14, 2020
Screening of a Custom-Designed Acid Fragment Library Identifies 1-Phenylpyrroles and 1-Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity
William Mahy, Mikesh Patel, David Steadman, et al.
ACS Chemical Neuroscience
|
June 22, 2022
Structural Analysis and Development of Notum Fragment Screening Hits
Yuguang Zhao, William Mahy, Nicky J Willis, et al.
Journal of Medicinal Chemistry
|
May 10, 2022
Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit
Nicky J Willis, William Mahy, James Sipthorp, et al.
Page
of 2