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Journal of Enzyme Inhibition and Medicinal Chemistry|March 18, 2026
Inhibition of prolyl-tRNA synthetase and efflux pumps as a dual-targeting strategy against multidrug-resistant bacteriaCristiane Tambascia, Jaqueline Cristina Silva, Barbara Carvalho Dos Reis, et al.Bioorganic Chemistry|August 28, 2021
Optimisation of 2-(N-phenyl carboxamide) triazolopyrimidine antimalarials with moderate to slow acting erythrocytic stage activityBrodie L Bailey, William Nguyen, Anna Ngo, et al.ACS Infectious Diseases|February 10, 2023
Fast-Killing Tyrosine Amide ((<i>S</i>)-SW228703) with Blood- and Liver-Stage Antimalarial Activity Associated with the Cyclic Amine Resistance Locus (<i>Pf</i>CARL)Leah S Imlay, Aloysus K Lawong, Suraksha Gahalawat, et al.Biorxiv : the Preprint Server for Biology|June 6, 2025
Identification of α-azacyclic acetamide-based inhibitors of <i>P. falciparum</i> Na <sup>+</sup> pump ( <i>Pf</i> ATP4) with fast-killing asexual blood-stage antimalarial activity by phenotypic screeningArturo Casas, Leah S Imlay, Vandana Thathy, et al.Antimicrobial Agents and Chemotherapy|July 25, 2025
Characterizing the quick-killing mechanism of action of azithromycin analogs against malaria parasitesEmma Y Mao, William Nguyen, Gouranga P Jana, et al.Parasites & Vectors|June 2, 2017
Assessing the anthelmintic activity of pyrazole-5-carboxamide derivatives against Haemonchus contortusYaqing Jiao, Sarah Preston, Hongjian Song, et al.ACS Infectious Diseases|September 8, 2025
Identification of α-Azacyclic Acetamide-Based Inhibitors of <i>P. falciparum</i> Na<sup>+</sup> Pump (<i>Pf</i>ATP4) with Fast-Killing Asexual Blood-Stage Antimalarial Activity by Phenotypic ScreeningArturo Casas, Leah S Imlay, Vandana Thathy, et al.Chemmedchem|September 21, 2022
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2Benoît Laleu, Kelly Rubiano, Tomas Yeo, et al.Journal of Medicinal Chemistry|August 26, 2021
Discovery and Structure-Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious AntimalarialsBenoît Laleu, Yuichiro Akao, Atsuko Ochida, et al.Journal of Medicinal Chemistry|February 23, 2021
Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in <i>Plasmodium falciparum</i>Aloysus Lawong, Suraksha Gahalawat, John Okombo, et al.Pageof 7