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Journal of Medicinal Chemistry|March 3, 2006
Microwave-accelerated synthesis of P1'-extended HIV-1 protease inhibitors encompassing a tertiary alcohol in the transition-state mimicking scaffoldJenny K Ekegren, Nina Ginman, Asa Johansson, et al.Bioorganic & Medicinal Chemistry|June 16, 2012
Highly potent macrocyclic BACE-1 inhibitors incorporating a hydroxyethylamine core: design, synthesis and X-ray crystal structures of enzyme inhibitor complexesVeronica Sandgren, Tatiana Agback, Per-Ola Johansson, et al.Bioorganic & Medicinal Chemistry|August 2, 2005
Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and IIDaniel Muthas, Daniel Nöteberg, Yogesh A Sabnis, et al.Bioorganic & Medicinal Chemistry|November 17, 2006
Synthesis of novel potent hepatitis C virus NS3 protease inhibitors: discovery of 4-hydroxy-cyclopent-2-ene-1,2-dicarboxylic acid as a N-acyl-L-hydroxyproline bioisostereFredrik Thorstensson, Fredrik Wångsell, Ingemar Kvarnström, et al.Bone|October 27, 2007
Cathepsin K inhibitors prevent matrix-derived growth factor degradation by human osteoclastsKaren Fuller, Kevin M Lawrence, Jade L Ross, et al.Bioorganic & Medicinal Chemistry|December 25, 2010
Investigation of α-phenylnorstatine and α-benzylnorstatine as transition state isostere motifs in the search for new BACE-1 inhibitorsFredrik Wångsell, Patrik Nordeman, Jonas Sävmarker, et al.Bioorganic & Medicinal Chemistry|May 6, 2006
Potent inhibitors of the hepatitis C virus NS3 protease: use of a novel P2 cyclopentane-derived templatePer-Ola Johansson, Marcus Bäck, Ingemar Kvarnström, et al.Bioorganic & Medicinal Chemistry|May 22, 2003
Acyl sulfonamides as potent protease inhibitors of the hepatitis C virus full-Length NS3 (protease-helicase/NTPase): a comparative study of different C-terminalsAnja Johansson, Anton Poliakov, Eva Akerblom, et al.Journal of Medicinal Chemistry|January 25, 2008
Two-carbon-elongated HIV-1 protease inhibitors with a tertiary-alcohol-containing transition-state mimicXiongyu Wu, Per Ohrngren, Jenny K Ekegren, et al.Journal of Medicinal Chemistry|June 25, 2005
Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin IIPer-Ola Johansson, Jimmy Lindberg, Michael J Blackman, et al.Pageof 7