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Bioorganic & Medicinal Chemistry|June 18, 2022
Defined stereoisomers of 2″-amino NAD<sup>+</sup> and their activity against human sirtuins and a bacterial (ADP-ribosyl) transferaseSarah Zähringer, Tobias Rumpf, Jelena Melesina, et al.Chemmedchem|May 26, 2012
Design, synthesis, and biological evaluation of 2-aminobenzanilide derivatives as potent and selective HDAC inhibitorsDiana A Stolfa, Angela Stefanachi, Julia M Gajer, et al.Chemmedchem|September 3, 2019
Structure-Based Screening of Tetrazolylhydrazide Inhibitors versus KDM4 Histone DemethylasesPiotr H Małecki, Nicole Rüger, Martin Roatsch, et al.Angewandte Chemie (International Ed. in English)|January 11, 2016
Structure-Based Development of an Affinity Probe for Sirtuin 2Matthias Schiedel, Tobias Rumpf, Berin Karaman, et al.Methods in Molecular Biology (Clifton, N.J.)|October 18, 2022
Synthesis, Biochemical, and Cellular Evaluation of HDAC6 Targeting Proteolysis Targeting ChimerasSalma Darwish, Tino Heimburg, Johannes Ridinger, et al.Oncotarget|March 10, 2015
The histone code reader SPIN1 controls RET signaling in liposarcomaHenriette Franz, Holger Greschik, Dominica Willmann, et al.Molecules (Basel, Switzerland)|February 15, 2018
Identification of Bichalcones as Sirtuin Inhibitors by Virtual Screening and In Vitro TestingBerin Karaman, Zayan Alhalabi, Sören Swyter, et al.Chemical Communications (Cambridge, England)|March 22, 2016
A quinone mediator drives oxidations catalysed by alcohol dehydrogenase-containing cell lysatesJulian Haas, Michael A Schätzle, Syed M Husain, et al.Chemmedchem|December 19, 2008
Pyridylalanine-containing hydroxamic acids as selective HDAC6 inhibitorsStefan Schäfer, Laura Saunders, Sonja Schlimme, et al.ACS Chemical Neuroscience|November 11, 2024
Aromatic Amino Acid Hydroxylases as Off-Targets of Histone Deacetylase InhibitorsAnne Baumann, Niklas Papenkordt, Dina Robaa, et al.Pageof 24