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Journal of Medicinal Chemistry|June 3, 2017
Design, Multicomponent Synthesis, and Anticancer Activity of a Focused Histone Deacetylase (HDAC) Inhibitor Library with Peptoid-Based Cap GroupsViktoria Krieger, Alexandra Hamacher, Christoph G W Gertzen, et al.European Journal of Medicinal Chemistry|August 15, 2021
Synthesis, structure-activity relationships, cocrystallization and cellular characterization of novel smHDAC8 inhibitors for the treatment of schistosomiasisEhab Ghazy, Tino Heimburg, Julien Lancelot, et al.Journal of Medicinal Chemistry|December 1, 2017
Structure-Based Design and Biological Characterization of Selective Histone Deacetylase 8 (HDAC8) Inhibitors with Anti-Neuroblastoma ActivityTino Heimburg, Fiona R Kolbinger, Patrik Zeyen, et al.Archiv Der Pharmazie|November 22, 2023
Quinoline-based thiazolyl-hydrazones target cancer cells through autophagy inhibitionVladimir Ćurčić, Mateusz Olszewski, Natalia Maciejewska, et al.ACS Infectious Diseases|October 31, 2019
Screening and Phenotypical Characterization of Schistosoma mansoni Histone Deacetylase 8 (SmHDAC8) Inhibitors as Multistage Antischistosomal AgentsFulvio Saccoccia, Margherita Brindisi, Roberto Gimmelli, et al.Journal of Medicinal Chemistry|January 16, 2019
Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 InhibitorsKatharina Vögerl, Nghia Ong, Johanna Senger, et al.Angewandte Chemie (International Ed. in English)|October 30, 2025
From Pharmacophore to Warhead: NAD+-Targeting Triazoles as Mechanism-Based Sirtuin InhibitorsFlorian Friedrich, Marat Meleshin, Niklas Papenkordt, et al.European Journal of Medicinal Chemistry|March 20, 2022
Identification of histone deacetylase 10 (HDAC10) inhibitors that modulate autophagy in transformed cellsPatrik Zeyen, Yanira Zeyn, Daniel Herp, et al.Chemmedchem|October 17, 2022
Chemically Diverse S. mansoni HDAC8 Inhibitors Reduce Viability in Worm Larval and Adult StagesBeatrice Noce, Elisabetta Di Bello, Clemens Zwergel, et al.International Journal of Molecular Sciences|June 2, 2021
Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 InhibitorsChiara Luise, Dina Robaa, Pierre Regenass, et al.Pageof 24