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Journal of Medicinal Chemistry|June 7, 2024
Structure-Activity Studies of 1,2,4-Oxadiazoles for the Inhibition of the NAD+-Dependent Lysine Deacylase Sirtuin 2Arianna Colcerasa, Florian Friedrich, Jelena Melesina, et al.European Journal of Medicinal Chemistry|November 17, 2020
Novel quinolone-based potent and selective HDAC6 inhibitors: Synthesis, molecular modeling studies and biological investigationNicola Relitti, A Prasanth Saraswati, Giulia Chemi, et al.Cell Death and Differentiation|March 9, 2018
A kinome-wide RNAi screen identifies ALK as a target to sensitize neuroblastoma cells for HDAC8-inhibitor treatmentJing Shen, Sara Najafi, Sina Stäble, et al.Plos Pathogens|October 3, 2013
Structural basis for the inhibition of histone deacetylase 8 (HDAC8), a key epigenetic player in the blood fluke Schistosoma mansoniMartin Marek, Srinivasaraghavan Kannan, Alexander-Thomas Hauser, et al.Nature Communications|February 13, 2015
Selective Sirt2 inhibition by ligand-induced rearrangement of the active siteTobias Rumpf, Matthias Schiedel, Berin Karaman, et al.Future Medicinal Chemistry|August 31, 2016
Tofacitinib and analogs as inhibitors of the histone kinase PRK1 (PKN1)Dmytro Ostrovskyi, Tobias Rumpf, Julia Eib, et al.Journal of Medicinal Chemistry|March 27, 2024
Discovery of a Potent, Selective, and Cell-Active SPIN1 InhibitorYan Xiong, Holger Greschik, Catrine Johansson, et al.Journal of Medicinal Chemistry|October 23, 2018
Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional DeterminantsMartin Marek, Tajith B Shaik, Tino Heimburg, et al.European Journal of Medicinal Chemistry|August 10, 2018
Novel spiroindoline HDAC inhibitors: Synthesis, molecular modelling and biological studiesMargherita Brindisi, Johanna Senger, Caterina Cavella, et al.Nature Structural & Molecular Biology|May 8, 2019
KMT9 monomethylates histone H4 lysine 12 and controls proliferation of prostate cancer cellsEric Metzger, Sheng Wang, Sylvia Urban, et al.Pageof 24