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European Journal of Medicinal Chemistry
|
September 19, 2014
Identification of two novel RET kinase inhibitors through MCR-based drug discovery: design, synthesis and evaluation
Brendan Frett, Marialuisa Moccia, Francesca Carlomagno, et al.
The AAPS Journal
|
December 20, 2019
Structural Characterization of the Aurora Kinase B "DFG-flip" Using Metadynamics
Naga Rajiv Lakkaniga, Meenakshisundaram Balasubramaniam, Shuxing Zhang, et al.
Medchemcomm
|
February 5, 2016
Identification of pyrazine-based TrkA inhibitors: design, synthesis, evaluation, and computational modeling studies
Brendan Frett, Nick McConnell, Yuanxiang Wang, et al.
Chemistryselect
|
August 25, 2018
Synthesis of Constrained Heterocycles Employing Two Post-Ugi Cyclization Methods for Rapid Library Generation with In Cellulo Activity
Nicholas McConnell, Zhigang Xu, Vishnu Kumarasamy, et al.
Chemmedchem
|
February 9, 2021
Pyrazoloadenine Inhibitors of the RET Lung Cancer Oncoprotein Discovered by a Fragment Optimization Approach
Debasmita Saha, Katie Rose Ryan, Naga Rajiv Lakkaniga, et al.
Journal of Medicinal Chemistry
|
September 25, 2019
The Exploration of Chirality for Improved Druggability within the Human Kinome
Debasmita Saha, Anupreet Kharbanda, Wei Yan, et al.
Journal of Medicinal Chemistry
|
February 13, 2014
Therapeutic melting pot of never in mitosis gene a related kinase 2 (Nek2): a perspective on Nek2 as an oncology target and recent advancements in Nek2 small molecule inhibition
Brendan Frett, Robert V Brown, Mingliang Ma, et al.
European Journal of Medicinal Chemistry
|
September 18, 2025
Discovery of novel 1H-pyrazolo[3,4-d]pyrimidine derivatives as BRK/PTK6 inhibitors
Baku Acharya, Maha Hanafi, Luke Enemark, et al.
European Journal of Medicinal Chemistry
|
August 22, 2021
Discovery of 4-aminoquinolines as highly selective TGFβR1 inhibitors with an attenuated MAP4K4 profile for potential applications in immuno-oncology
Anupreet Kharbanda, Phuc Tran, Lingtian Zhang, et al.
European Journal of Medicinal Chemistry
|
July 28, 2020
Discovery of SP-96, the first non-ATP-competitive Aurora Kinase B inhibitor, for reduced myelosuppression
Naga Rajiv Lakkaniga, Lingtian Zhang, Binyam Belachew, et al.
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of 6
Search research articles
Search
Showing results (11-20 of 54) with videos related to
Sort By:
Page
of 6
European Journal of Medicinal Chemistry
|
September 19, 2014
Identification of two novel RET kinase inhibitors through MCR-based drug discovery: design, synthesis and evaluation
Brendan Frett, Marialuisa Moccia, Francesca Carlomagno, et al.
The AAPS Journal
|
December 20, 2019
Structural Characterization of the Aurora Kinase B "DFG-flip" Using Metadynamics
Naga Rajiv Lakkaniga, Meenakshisundaram Balasubramaniam, Shuxing Zhang, et al.
Medchemcomm
|
February 5, 2016
Identification of pyrazine-based TrkA inhibitors: design, synthesis, evaluation, and computational modeling studies
Brendan Frett, Nick McConnell, Yuanxiang Wang, et al.
Chemistryselect
|
August 25, 2018
Synthesis of Constrained Heterocycles Employing Two Post-Ugi Cyclization Methods for Rapid Library Generation with In Cellulo Activity
Nicholas McConnell, Zhigang Xu, Vishnu Kumarasamy, et al.
Chemmedchem
|
February 9, 2021
Pyrazoloadenine Inhibitors of the RET Lung Cancer Oncoprotein Discovered by a Fragment Optimization Approach
Debasmita Saha, Katie Rose Ryan, Naga Rajiv Lakkaniga, et al.
Journal of Medicinal Chemistry
|
September 25, 2019
The Exploration of Chirality for Improved Druggability within the Human Kinome
Debasmita Saha, Anupreet Kharbanda, Wei Yan, et al.
Journal of Medicinal Chemistry
|
February 13, 2014
Therapeutic melting pot of never in mitosis gene a related kinase 2 (Nek2): a perspective on Nek2 as an oncology target and recent advancements in Nek2 small molecule inhibition
Brendan Frett, Robert V Brown, Mingliang Ma, et al.
European Journal of Medicinal Chemistry
|
September 18, 2025
Discovery of novel 1H-pyrazolo[3,4-d]pyrimidine derivatives as BRK/PTK6 inhibitors
Baku Acharya, Maha Hanafi, Luke Enemark, et al.
European Journal of Medicinal Chemistry
|
August 22, 2021
Discovery of 4-aminoquinolines as highly selective TGFβR1 inhibitors with an attenuated MAP4K4 profile for potential applications in immuno-oncology
Anupreet Kharbanda, Phuc Tran, Lingtian Zhang, et al.
European Journal of Medicinal Chemistry
|
July 28, 2020
Discovery of SP-96, the first non-ATP-competitive Aurora Kinase B inhibitor, for reduced myelosuppression
Naga Rajiv Lakkaniga, Lingtian Zhang, Binyam Belachew, et al.
Page
of 6