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Journal of Biomolecular Screening|February 13, 2014
Small-Molecule Library Subset Screening as an Aid for Accelerating Lead IdentificationMaureen H Beresini, Yichin Liu, Timothy D Dawes, et al.Journal of Laboratory Automation|June 17, 2015
Compound Transfer by Acoustic Droplet Ejection Promotes Quality and Efficiency in Ultra-High-Throughput Screening CampaignsTimothy D Dawes, Rebecca Turincio, Steven W Jones, et al.ACS Medicinal Chemistry Letters|March 18, 2016
Development of a Potent, Specific CDK8 Kinase Inhibitor Which Phenocopies CDK8/19 Knockout CellsMichael F T Koehler, Philippe Bergeron, Elizabeth M Blackwood, et al.ACS Medicinal Chemistry Letters|December 18, 2020
Identification of BRaf-Sparing Amino-Thienopyrimidines with Potent IRE1α Inhibitory ActivityRamsay E Beveridge, Heidi Ackerly Wallweber, Avi Ashkenazi, et al.Nature Communications|December 15, 2020
Activation of the IRE1 RNase through remodeling of the kinase front pocket by ATP-competitive ligandsElena Ferri, Adrien Le Thomas, Heidi Ackerly Wallweber, et al.Journal of Medicinal Chemistry|May 15, 2024
Discovery of Potent, Selective, and Orally Available IRE1α Inhibitors Demonstrating Comparable PD Modulation to IRE1 Knockdown in a Multiple Myeloma ModelMarie-Gabrielle Braun, Avi Ashkenazi, Ramsay E Beveridge, et al.Journal of Medicinal Chemistry|November 21, 2017
A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) InhibitorsSarah M Bronner, Jeremy Murray, F Anthony Romero, et al.Science (New York, N.Y.)|December 19, 2015
Structural basis of Nav1.7 inhibition by an isoform-selective small-molecule antagonistShivani Ahuja, Susmith Mukund, Lunbin Deng, et al.Bioorganic & Medicinal Chemistry Letters|November 13, 2024
Discovery of potent dihydro-oxazinoquinolinone inhibitors of GuaB for the treatment of tuberculosisYuebiao Zhou, Ignacio Aliagas, Shumei Wang, et al.Nature|October 19, 2017
USP7 small-molecule inhibitors interfere with ubiquitin bindingLorna Kategaya, Paola Di Lello, Lionel Rougé, et al.Pageof 5