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Journal of Medicinal Chemistry|March 1, 2022
Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting Blood-Stage Antimalarial with a High Barrier to Resistance and Potential for Single-Dose Cures in Uncomplicated MalariaBenjamin R Taft, Fumiaki Yokokawa, Tom Kirrane, et al.Elife|September 30, 2025
A drug repurposing approach reveals targetable epigenetic pathways in <i>Plasmodium vivax</i> hypnozoitesSteven P Maher, Malina A Bakowski, Amélie Vantaux, et al.Nature Communications|April 21, 2022
Preclinical characterization and target validation of the antimalarial pantothenamide MMV693183Laura E de Vries, Patrick A M Jansen, Catalina Barcelo, et al.Science Translational Medicine|July 17, 2015
A long-duration dihydroorotate dehydrogenase inhibitor (DSM265) for prevention and treatment of malariaMargaret A Phillips, Julie Lotharius, Kennan Marsh, et al.Research Square|December 9, 2024
Revisiting the Plasmodium falciparum druggable genome using predicted structures and data miningKarla P Godinez-Macias, Daisy Chen, J Lincoln Wallis, et al.NPJ Drug Discovery|March 11, 2025
Revisiting the <i>Plasmodium falciparum</i> druggable genome using predicted structures and data miningKarla P Godinez-Macias, Daisy Chen, J Lincoln Wallis, et al.Nature Communications|May 25, 2017
A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistancePaul M O'Neill, Richard K Amewu, Susan A Charman, et al.Science Translational Medicine|April 28, 2017
Antimalarial efficacy of MMV390048, an inhibitor of <i>Plasmodium</i> phosphatidylinositol 4-kinaseTanya Paquet, Claire Le Manach, Diego González Cabrera, et al.Nature|June 19, 2015
A novel multiple-stage antimalarial agent that inhibits protein synthesisBeatriz Baragaña, Irene Hallyburton, Marcus C S Lee, et al.Pageof 6