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Celine Valant

Showing results (11-20 of 73) with videos related to

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Bioorganic & Medicinal Chemistry Letters|May 27, 2011
The synthesis and biological evaluation of 2-amino-4,5,6,7,8,9-hexahydrocycloocta[b]thiophenes as allosteric modulators of the A1 adenosine receptorLuigi Aurelio, Arthur Christopoulos, Bernard L Flynn, et al.
Journal of Medicinal Chemistry|May 31, 2013
Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptorShailesh N Mistry, Celine Valant, Patrick M Sexton, et al.
Endocrinology|January 3, 2012
Positive and negative allosteric modulators promote biased signaling at the calcium-sensing receptorAnna E Davey, Katie Leach, Celine Valant, et al.
Journal of Medicinal Chemistry|June 12, 2009
Allosteric modulators of the adenosine A1 receptor: synthesis and pharmacological evaluation of 4-substituted 2-amino-3-benzoylthiophenesLuigi Aurelio, Celine Valant, Bernard L Flynn, et al.
Bioorganic & Medicinal Chemistry Letters|March 3, 2012
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT₂C agonistsRichard J Conway, Celine Valant, Arthur Christopoulos, et al.
Science Advances|September 11, 2024
Positive allosteric modulation of a GPCR ternary complexWessel A C Burger, Christopher J Draper-Joyce, Celine Valant, et al.
Molecular Pharmacology|May 28, 2011
Polymorphism and ligand dependent changes in human glucagon-like peptide-1 receptor (GLP-1R) function: allosteric rescue of loss of function mutationCassandra Koole, Denise Wootten, John Simms, et al.
Molecular Pharmacology|June 16, 2010
Delineating the mode of action of adenosine A1 receptor allosteric modulatorsCeline Valant, Luigi Aurelio, Vijay B Urmaliya, et al.
FASEB Journal : Official Publication of the Federation of American Societies for Experimental Biology|March 21, 2007
A novel, conformation-specific allosteric inhibitor of the tachykinin NK2 receptor (NK2R) with functionally selective propertiesEmeline L Maillet, Nadia Pellegrini, Celine Valant, et al.
Molecular Pharmacology|June 27, 2013
Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M₁ muscarinic acetylcholine receptorPeter Keov, Celine Valant, Shane M Devine, et al.
Pageof 8

Showing results (11-20 of 73) with videos related to

Sort By:
Pageof 8
Bioorganic & Medicinal Chemistry Letters|May 27, 2011
The synthesis and biological evaluation of 2-amino-4,5,6,7,8,9-hexahydrocycloocta[b]thiophenes as allosteric modulators of the A1 adenosine receptorLuigi Aurelio, Arthur Christopoulos, Bernard L Flynn, et al.
Journal of Medicinal Chemistry|May 31, 2013
Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptorShailesh N Mistry, Celine Valant, Patrick M Sexton, et al.
Endocrinology|January 3, 2012
Positive and negative allosteric modulators promote biased signaling at the calcium-sensing receptorAnna E Davey, Katie Leach, Celine Valant, et al.
Journal of Medicinal Chemistry|June 12, 2009
Allosteric modulators of the adenosine A1 receptor: synthesis and pharmacological evaluation of 4-substituted 2-amino-3-benzoylthiophenesLuigi Aurelio, Celine Valant, Bernard L Flynn, et al.
Bioorganic & Medicinal Chemistry Letters|March 3, 2012
Synthesis and SAR study of 4-arylpiperidines and 4-aryl-1,2,3,6-tetrahydropyridines as 5-HT₂C agonistsRichard J Conway, Celine Valant, Arthur Christopoulos, et al.
Science Advances|September 11, 2024
Positive allosteric modulation of a GPCR ternary complexWessel A C Burger, Christopher J Draper-Joyce, Celine Valant, et al.
Molecular Pharmacology|May 28, 2011
Polymorphism and ligand dependent changes in human glucagon-like peptide-1 receptor (GLP-1R) function: allosteric rescue of loss of function mutationCassandra Koole, Denise Wootten, John Simms, et al.
Molecular Pharmacology|June 16, 2010
Delineating the mode of action of adenosine A1 receptor allosteric modulatorsCeline Valant, Luigi Aurelio, Vijay B Urmaliya, et al.
FASEB Journal : Official Publication of the Federation of American Societies for Experimental Biology|March 21, 2007
A novel, conformation-specific allosteric inhibitor of the tachykinin NK2 receptor (NK2R) with functionally selective propertiesEmeline L Maillet, Nadia Pellegrini, Celine Valant, et al.
Molecular Pharmacology|June 27, 2013
Reverse engineering of the selective agonist TBPB unveils both orthosteric and allosteric modes of action at the M₁ muscarinic acetylcholine receptorPeter Keov, Celine Valant, Shane M Devine, et al.
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