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Celine Valant

Showing results (21-30 of 73) with videos related to

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Proceedings of the National Academy of Sciences of the United States of America|September 8, 2016
Accelerated structure-based design of chemically diverse allosteric modulators of a muscarinic G protein-coupled receptorYinglong Miao, Dahlia Anne Goldfeld, Ee Von Moo, et al.
Journal of Medicinal Chemistry|September 3, 2010
Effects of conformational restriction of 2-amino-3-benzoylthiophenes on A(1) adenosine receptor modulationLuigi Aurelio, Celine Valant, Bernard L Flynn, et al.
British Journal of Pharmacology|December 23, 2022
Importance of receptor expression in the classification of novel ligands at the M<sub>2</sub> muscarinic acetylcholine receptorYe Jiang, Mahmuda Yeasmin, Arisbel B Gondin, et al.
Journal of Medicinal Chemistry|May 27, 2014
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M ₁ muscarinic acetylcholine receptorBriana J Davie, Celine Valant, Jonathan M White, et al.
ACS Chemical Neuroscience|December 14, 2021
Structural Features of Iperoxo-BQCA Muscarinic Acetylcholine Receptor Hybrid Ligands Determining Subtype Selectivity and EfficacyMatthew C L Wakeham, Briana J Davie, David K Chalmers, et al.
Bioorganic & Medicinal Chemistry|September 16, 2009
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonistsLuigi Aurelio, Celine Valant, Heidi Figler, et al.
The Journal of Biological Chemistry|August 30, 2008
A novel mechanism of G protein-coupled receptor functional selectivity. Muscarinic partial agonist McN-A-343 as a bitopic orthosteric/allosteric ligandCeline Valant, Karen J Gregory, Nathan E Hall, et al.
Molecular Pharmacology|June 22, 2023
Role of Conserved Tyrosine Lid Residues in the Activation of the M<sub>2</sub> Muscarinic Acetylcholine ReceptorVi Pham, Maria Clazina Cornelia Habben Jansen, Geoff Thompson, et al.
The Journal of Biological Chemistry|July 10, 2014
Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptorPeter Keov, Laura López, Shane M Devine, et al.
Journal of Medicinal Chemistry|September 13, 2022
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ<i>-</i>Opioid ReceptorOwindeep Deo, Sadia Alvi, Vi Pham, et al.
Pageof 8

Showing results (21-30 of 73) with videos related to

Sort By:
Pageof 8
Proceedings of the National Academy of Sciences of the United States of America|September 8, 2016
Accelerated structure-based design of chemically diverse allosteric modulators of a muscarinic G protein-coupled receptorYinglong Miao, Dahlia Anne Goldfeld, Ee Von Moo, et al.
Journal of Medicinal Chemistry|September 3, 2010
Effects of conformational restriction of 2-amino-3-benzoylthiophenes on A(1) adenosine receptor modulationLuigi Aurelio, Celine Valant, Bernard L Flynn, et al.
British Journal of Pharmacology|December 23, 2022
Importance of receptor expression in the classification of novel ligands at the M<sub>2</sub> muscarinic acetylcholine receptorYe Jiang, Mahmuda Yeasmin, Arisbel B Gondin, et al.
Journal of Medicinal Chemistry|May 27, 2014
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M ₁ muscarinic acetylcholine receptorBriana J Davie, Celine Valant, Jonathan M White, et al.
ACS Chemical Neuroscience|December 14, 2021
Structural Features of Iperoxo-BQCA Muscarinic Acetylcholine Receptor Hybrid Ligands Determining Subtype Selectivity and EfficacyMatthew C L Wakeham, Briana J Davie, David K Chalmers, et al.
Bioorganic & Medicinal Chemistry|September 16, 2009
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonistsLuigi Aurelio, Celine Valant, Heidi Figler, et al.
The Journal of Biological Chemistry|August 30, 2008
A novel mechanism of G protein-coupled receptor functional selectivity. Muscarinic partial agonist McN-A-343 as a bitopic orthosteric/allosteric ligandCeline Valant, Karen J Gregory, Nathan E Hall, et al.
Molecular Pharmacology|June 22, 2023
Role of Conserved Tyrosine Lid Residues in the Activation of the M<sub>2</sub> Muscarinic Acetylcholine ReceptorVi Pham, Maria Clazina Cornelia Habben Jansen, Geoff Thompson, et al.
The Journal of Biological Chemistry|July 10, 2014
Molecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptorPeter Keov, Laura López, Shane M Devine, et al.
Journal of Medicinal Chemistry|September 13, 2022
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ<i>-</i>Opioid ReceptorOwindeep Deo, Sadia Alvi, Vi Pham, et al.
Pageof 8