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Journal of Medicinal Chemistry
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August 22, 2024
The Missing Link(er): A Roadmap to Macrocyclization in Drug Discovery
Christian Brudy, Carlo Walz, Moritz Spiske, et al.
Angewandte Chemie (International Ed. in English)
|
January 3, 2025
Conformationally Restricted Macrocycles as Improved FKBP51 Inhibitors Enabled by Systematic Linker Derivatization
Moritz Spiske, Christian Meyners, Michael Bauder, et al.
Angewandte Chemie (International Ed. in English)
|
January 3, 2025
Conformational Plasticity and Binding Affinity Enhancement Controlled by Linker Derivatization in Macrocycles
Vanessa Buffa, Carlo Walz, Christian Meyners, et al.
Journal of Medicinal Chemistry
|
November 22, 2025
Linker Modification Enables Control of Key Functional Group Orientation in Macrocycles
Christian Brudy, Enrico Ruijsenaars, Christian Meyners, et al.
Page
of 1
Search research articles
Search
Showing results (1-10 of 4) with videos related to
Sort By:
Page
of 1
Journal of Medicinal Chemistry
|
August 22, 2024
The Missing Link(er): A Roadmap to Macrocyclization in Drug Discovery
Christian Brudy, Carlo Walz, Moritz Spiske, et al.
Angewandte Chemie (International Ed. in English)
|
January 3, 2025
Conformationally Restricted Macrocycles as Improved FKBP51 Inhibitors Enabled by Systematic Linker Derivatization
Moritz Spiske, Christian Meyners, Michael Bauder, et al.
Angewandte Chemie (International Ed. in English)
|
January 3, 2025
Conformational Plasticity and Binding Affinity Enhancement Controlled by Linker Derivatization in Macrocycles
Vanessa Buffa, Carlo Walz, Christian Meyners, et al.
Journal of Medicinal Chemistry
|
November 22, 2025
Linker Modification Enables Control of Key Functional Group Orientation in Macrocycles
Christian Brudy, Enrico Ruijsenaars, Christian Meyners, et al.
Page
of 1