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Bioorganic & Medicinal Chemistry Letters|May 5, 2021
Design and evaluation of 1,2,3-dithiazoles and fused 1,2,4-dithiazines as anti-cancer agentsKaitlyn A Maffuid, Maria Koyioni, Chad D Torrice, et al.Bioorganic & Medicinal Chemistry Letters|February 24, 2015
Novel fused tetrathiocines as antivirals that target the nucleocapsid zinc finger containing protein of the feline immunodeficiency virus (FIV) as a model of HIV infectionChristopher R M Asquith, Marina L Meli, Lidia S Konstantinova, et al.British Journal of Pharmacology|February 27, 2025
Chemosensory signalling in human sperm is controlled by Ca2+ influx via CatSper and Ca2+ clearance via plasma membrane Ca2+ ATPasesLeonie Herrmann, Christoph Brenker, Teresa Mittermair, et al.Antimicrobial Agents and Chemotherapy|October 16, 2019
Quinazoline-Based Antivirulence Compounds Selectively Target Salmonella PhoP/PhoQ Signal Transduction SystemMaría Ayelén Carabajal, Christopher R M Asquith, Tuomo Laitinen, et al.Scientific Reports|March 1, 2024
Enhancing colistin efficacy against Salmonella infections with a quinazoline-based dual therapeutic strategyCarlos A Lobertti, Fernán O Gizzi, Christian Magni, et al.Antibiotics (Basel, Switzerland)|December 11, 2019
Synthesis and Identification of Pentathiepin-Based Inhibitors of Sporothrix brasiliensisChristopher R M Asquith, Ana C S Machado, Luisa H M de Miranda, et al.Chemmedchem|May 29, 2018
Synthesis and Pharmacological Evaluation of Enantiomerically Pure GluN2B Selective NMDA Receptor AntagonistsFrederik Börgel, Marina Szermerski, Julian A Schreiber, et al.Journal of Medicinal Chemistry|July 15, 2021
Hinge Binder Scaffold Hopping Identifies Potent Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CAMKK2) Inhibitor ChemotypesBenjamin J Eduful, Sean N O'Byrne, Louisa Temme, et al.Bioorganic & Medicinal Chemistry Letters|May 13, 2014
Evaluation of the antiviral efficacy of bis[1,2]dithiolo[1,4]thiazines and bis[1,2]dithiolopyrrole derivatives against the nucelocapsid protein of the Feline Immunodeficiency Virus (FIV) as a model for HIV infectionChristopher R M Asquith, Marina L Meli, Lidia S Konstantinova, et al.Bioorganic Chemistry|May 8, 2026
4-Anilinoquinazoline carbamate derivatization as a platform for prodrug design and localized drug deliveryMabel Barreiro Carpio, Coleman D Walker, Audrey Fikes, et al.Pageof 6