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Acta Chimica Slovenica|September 25, 2013
New Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones Fluoroderivatives as Human A1 Adenosine Receptor LigandsAlessia Graziano, Maria Paola Giovannoni, Agostino Cilibrizzi, et al.
Journal of Medicinal Chemistry|July 13, 2013
Optimization of N-benzoylindazole derivatives as inhibitors of human neutrophil elastaseLetizia Crocetti, Igor A Schepetkin, Agostino Cilibrizzi, et al.
Rheumatology (Oxford, England)|April 2, 2016
Effects of the neutrophil elastase inhibitor EL-17 in rat adjuvant-induced arthritisLorenzo Di Cesare Mannelli, Laura Micheli, Lorenzo Cinci, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|January 18, 2003
Synthesis and evaluation of some pyrazolo[3,4-d]pyridazinones and analogues as PDE 5 inhibitors potentially useful as peripheral vasodilator agentsVittorio Dal Piaz, Maria Carla Castellana, Claudia Vergelli, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|July 22, 2015
Cinnoline derivatives as human neutrophil elastase inhibitorsMaria Paola Giovannoni, Igor A Schepetkin, Letizia Crocetti, et al.
Drug Development Research|April 20, 2019
Further modifications of 1H-pyrrolo[2,3-b]pyridine derivatives as inhibitors of human neutrophil elastaseMaria P Giovannoni, Niccolò Cantini, Letizia Crocetti, et al.
Pharmaceuticals (Basel, Switzerland)|November 10, 2022
Ligand Growing Experiments Suggested 4-amino and 4-ureido pyridazin-3(2<i>H</i>)-one as Novel Scaffold for FABP4 InhibitionLetizia Crocetti, Giuseppe Floresta, Chiara Zagni, et al.
Bioorganic & Medicinal Chemistry Letters|September 26, 2021
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitorsNiccolo Cantini, Letizia Crocetti, Gabriella Guerrini, et al.
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