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Bioorganic & Medicinal Chemistry|July 12, 2011
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastaseLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.Bioorganic & Medicinal Chemistry|November 3, 2018
1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitorsLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|June 15, 2017
Isoxazol-5(2H)-one: a new scaffold for potent human neutrophil elastase (HNE) inhibitorsClaudia Vergelli, Igor A Schepetkin, Letizia Crocetti, et al.Bioorganic & Medicinal Chemistry|November 21, 2020
Exploration of nitrogen heterocycle scaffolds for the development of potent human neutrophil elastase inhibitorsNiccolò Cantini, Andrei I Khlebnikov, Letizia Crocetti, et al.Bioorganic & Medicinal Chemistry|May 22, 2012
Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonistsAgostino Cilibrizzi, Igor A Schepetkin, Gianluca Bartolucci, et al.Drug Development Research|July 31, 2016
Synthesis and Pharmacological Evaluation of Indole Derivatives as Deaza Analogues of Potent Human Neutrophil Elastase InhibitorsLetizia Crocetti, Igor A Schepetkin, Giovanna Ciciani, et al.Chemistry Central Journal|December 8, 2017
Synthesis and analytical characterization of new thiazol-2-(3H)-ones as human neutrophil elastase (HNE) inhibitorsLetizia Crocetti, Gianluca Bartolucci, Agostino Cilibrizzi, et al.Molecules (Basel, Switzerland)|February 27, 2026
Discovery of Potent PDE4 Inhibitors with 3(2H)-Pyridazinone Scaffold: Synthesis, In Silico Studies and In Vitro/Vivo EvaluationClaudia Vergelli, Letizia Crocetti, Gabriella Guerrini, et al.Bioorganic & Medicinal Chemistry|October 13, 2010
Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligandsMaria Paola Giovannoni, Claudia Vergelli, Agostino Cilibrizzi, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|July 5, 2018
Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitorsMaria Paola Giovannoni, Igor A Schepetkin, Mark T Quinn, et al.Pageof 6