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Cerebrovascular Diseases Extra
|
May 1, 2019
Nonsteroidal Anti-Inflammatory Drugs: A Potential Pharmacological Treatment for Intracranial Aneurysm
Courtney L Fisher, Stacie L Demel
Journal of Hypertension
|
August 9, 2022
Mineralocorticoid receptor antagonism improves transient receptor potential vanilloid 4-dependent dilation of cerebral parenchymal arterioles and cognition in a genetic model of hypertension
Laura C Chambers, Janice M Diaz-Otero, Courtney L Fisher, et al.
Journal of Medicinal Chemistry
|
November 11, 2022
Structure-Activity Studies of 1<i>H</i>-Imidazo[4,5-<i>c</i>]quinolin-4-amine Derivatives as A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulators
Lucas B Fallot, R Rama Suresh, Courtney L Fisher, et al.
ACS Pharmacology & Translational Science
|
September 14, 2023
First Potent Macrocyclic A<sub>3</sub> Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences
Dilip K Tosh, Courtney L Fisher, Veronica Salmaso, et al.
Molecular Pharmacology
|
January 5, 2024
Extrahelical Binding Site for a 1<i>H</i>-Imidazo[4,5-c]quinolin-4-amine A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7
Courtney L Fisher, Matteo Pavan, Veronica Salmaso, et al.
Journal of Medicinal Chemistry
|
April 10, 2020
Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A<sub>3</sub> Adenosine Receptors: Affinity Enhancement by <i>N</i><sup>6</sup>-(2-Phenylethyl) Substitution
Dilip K Tosh, Veronica Salmaso, Harsha Rao, et al.
ACS Pharmacology & Translational Science
|
August 19, 2022
Characterization of Dual-Acting A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulators That Preferentially Enhance Adenosine-Induced Gα<sub>i3</sub> and Gα<sub>oA</sub> Isoprotein Activation
Courtney L Fisher, Lucas B Fallot, Tina C Wan, et al.
Journal of Medicinal Chemistry
|
July 3, 2024
Lipid Trolling to Optimize A<sub>3</sub> Adenosine Receptor-Positive Allosteric Modulators (PAMs)
Balaram Pradhan, Matteo Pavan, Courtney L Fisher, et al.
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Showing results (1-10 of 8) with videos related to
Sort By:
Page
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Cerebrovascular Diseases Extra
|
May 1, 2019
Nonsteroidal Anti-Inflammatory Drugs: A Potential Pharmacological Treatment for Intracranial Aneurysm
Courtney L Fisher, Stacie L Demel
Journal of Hypertension
|
August 9, 2022
Mineralocorticoid receptor antagonism improves transient receptor potential vanilloid 4-dependent dilation of cerebral parenchymal arterioles and cognition in a genetic model of hypertension
Laura C Chambers, Janice M Diaz-Otero, Courtney L Fisher, et al.
Journal of Medicinal Chemistry
|
November 11, 2022
Structure-Activity Studies of 1<i>H</i>-Imidazo[4,5-<i>c</i>]quinolin-4-amine Derivatives as A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulators
Lucas B Fallot, R Rama Suresh, Courtney L Fisher, et al.
ACS Pharmacology & Translational Science
|
September 14, 2023
First Potent Macrocyclic A<sub>3</sub> Adenosine Receptor Agonists Reveal G-Protein and β-Arrestin2 Signaling Preferences
Dilip K Tosh, Courtney L Fisher, Veronica Salmaso, et al.
Molecular Pharmacology
|
January 5, 2024
Extrahelical Binding Site for a 1<i>H</i>-Imidazo[4,5-c]quinolin-4-amine A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7
Courtney L Fisher, Matteo Pavan, Veronica Salmaso, et al.
Journal of Medicinal Chemistry
|
April 10, 2020
Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A<sub>3</sub> Adenosine Receptors: Affinity Enhancement by <i>N</i><sup>6</sup>-(2-Phenylethyl) Substitution
Dilip K Tosh, Veronica Salmaso, Harsha Rao, et al.
ACS Pharmacology & Translational Science
|
August 19, 2022
Characterization of Dual-Acting A<sub>3</sub> Adenosine Receptor Positive Allosteric Modulators That Preferentially Enhance Adenosine-Induced Gα<sub>i3</sub> and Gα<sub>oA</sub> Isoprotein Activation
Courtney L Fisher, Lucas B Fallot, Tina C Wan, et al.
Journal of Medicinal Chemistry
|
July 3, 2024
Lipid Trolling to Optimize A<sub>3</sub> Adenosine Receptor-Positive Allosteric Modulators (PAMs)
Balaram Pradhan, Matteo Pavan, Courtney L Fisher, et al.
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