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Biorxiv : the Preprint Server for Biology
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March 10, 2025
Prospective evaluation of structure-based simulations reveal their ability to predict the impact of kinase mutations on inhibitor binding
Sukrit Singh, Vytautas Gapsys, Matteo Aldeghi, et al.
Practical Radiation Oncology
|
January 18, 2024
Systematic Implementation of Effective Quality Assurance Processes for the Assessment of Radiation Target Volumes in Head and Neck Cancer
E Gogineni, D Schaefer, A Ewing, et al.
Journal of Medicinal Chemistry
|
October 5, 2001
Design and synthesis of a series of (2R)-N(4)-hydroxy-2-(3-hydroxybenzyl)-N(1)- [(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide derivatives as potent, selective, and orally bioavailable aggrecanase inhibitors
W Yao, Z R Wasserman, M Chao, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
July 28, 2007
Pharmacokinetics and pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a potent and selective inhibitor of tumor necrosis factor alpha-converting enzyme in rodents, dogs, chimpanzees, and humans
Mingxin Qian, Stephen A Bai, Bernice Brogdon, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 6, 2007
A new 4-(2-methylquinolin-4-ylmethyl)phenyl P1' group for the beta-amino hydroxamic acid derived TACE inhibitors
Xiao-Tao Chen, Bahman Ghavimi, Ronald L Corbett, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 27, 2003
Potent and selective aggrecanase inhibitors containing cyclic P1 substituents
Robert J Cherney, Ruowei Mo, Dayton T Meyer, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2003
Rational design, synthesis and structure-activity relationships of a cyclic succinate series of TNF-alpha converting enzyme inhibitors. Part 2: lead optimization
Chu-Biao Xue, Xiaohua He, John Roderick, et al.
Cellular Oncology (Dordrecht, Netherlands)
|
January 25, 2021
The potent AMPK inhibitor BAY-3827 shows strong efficacy in androgen-dependent prostate cancer models
Clara Lemos, Volker K Schulze, Simon J Baumgart, et al.
Journal of Medicinal Chemistry
|
October 26, 2021
Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A
Lars Wortmann, Nico Bräuer, Simon J Holton, et al.
Current Topics in Medicinal Chemistry
|
April 8, 2011
G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey
Nicole A Kratochwil, Silvia Gatti-McArthur, Marius C Hoener, et al.
Page
of 12
Search research articles
Search
Showing results (101-110 of 120) with videos related to
Sort By:
Page
of 12
Biorxiv : the Preprint Server for Biology
|
March 10, 2025
Prospective evaluation of structure-based simulations reveal their ability to predict the impact of kinase mutations on inhibitor binding
Sukrit Singh, Vytautas Gapsys, Matteo Aldeghi, et al.
Practical Radiation Oncology
|
January 18, 2024
Systematic Implementation of Effective Quality Assurance Processes for the Assessment of Radiation Target Volumes in Head and Neck Cancer
E Gogineni, D Schaefer, A Ewing, et al.
Journal of Medicinal Chemistry
|
October 5, 2001
Design and synthesis of a series of (2R)-N(4)-hydroxy-2-(3-hydroxybenzyl)-N(1)- [(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide derivatives as potent, selective, and orally bioavailable aggrecanase inhibitors
W Yao, Z R Wasserman, M Chao, et al.
Drug Metabolism and Disposition: the Biological Fate of Chemicals
|
July 28, 2007
Pharmacokinetics and pharmacodynamics of DPC 333 ((2R)-2-((3R)-3-amino-3{4-[2-methyl-4-quinolinyl) methoxy] phenyl}-2-oxopyrrolidinyl)-N-hydroxy-4-methylpentanamide)), a potent and selective inhibitor of tumor necrosis factor alpha-converting enzyme in rodents, dogs, chimpanzees, and humans
Mingxin Qian, Stephen A Bai, Bernice Brogdon, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 6, 2007
A new 4-(2-methylquinolin-4-ylmethyl)phenyl P1' group for the beta-amino hydroxamic acid derived TACE inhibitors
Xiao-Tao Chen, Bahman Ghavimi, Ronald L Corbett, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 27, 2003
Potent and selective aggrecanase inhibitors containing cyclic P1 substituents
Robert J Cherney, Ruowei Mo, Dayton T Meyer, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2003
Rational design, synthesis and structure-activity relationships of a cyclic succinate series of TNF-alpha converting enzyme inhibitors. Part 2: lead optimization
Chu-Biao Xue, Xiaohua He, John Roderick, et al.
Cellular Oncology (Dordrecht, Netherlands)
|
January 25, 2021
The potent AMPK inhibitor BAY-3827 shows strong efficacy in androgen-dependent prostate cancer models
Clara Lemos, Volker K Schulze, Simon J Baumgart, et al.
Journal of Medicinal Chemistry
|
October 26, 2021
Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A
Lars Wortmann, Nico Bräuer, Simon J Holton, et al.
Current Topics in Medicinal Chemistry
|
April 8, 2011
G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey
Nicole A Kratochwil, Silvia Gatti-McArthur, Marius C Hoener, et al.
Page
of 12