Search research articles
Contact Us
Filters
Showing results (431-440 of 459) with videos related to
Page
of 46
Sort By:
Bioorganic & Medicinal Chemistry Letters
|
December 22, 2005
Potent 2-[(pyrimidin-4-yl)amine}-1,3-thiazole-5-carbonitrile-based inhibitors of VEGFR-2 (KDR) kinase
John T Sisko, Thomas J Tucker, Mark T Bilodeau, et al.
Cancer Research
|
December 26, 2001
Evaluation of farnesyl:protein transferase and geranylgeranyl:protein transferase inhibitor combinations in preclinical models
R B Lobell, C A Omer, M T Abrams, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 12, 2001
Non-peptide alpha(v)beta(3) antagonists. Part 3: identification of potent RGD mimetics incorporating novel beta-amino acids as aspartic acid replacements
Paul J Coleman, Karen M Brashear, Cecilia A Hunt, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 28, 2006
Kinesin spindle protein (KSP) inhibitors. Part 2: the design, synthesis, and characterization of 2,4-diaryl-2,5-dihydropyrrole inhibitors of the mitotic kinesin KSP
Mark E Fraley, Robert M Garbaccio, Kenneth L Arrington, et al.
ACS Medicinal Chemistry Letters
|
June 6, 2014
Discovery of 4,4-Disubstituted Quinazolin-2-ones as T-Type Calcium Channel Antagonists
James C Barrow, Kenneth E Rittle, Thomas S Reger, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 30, 2017
Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics
Scott E Wolkenberg, M Brad Nolt, Mark T Bilodeau, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 1, 2007
Kinesin spindle protein (KSP) inhibitors. Part 6: Design and synthesis of 3,5-diaryl-4,5-dihydropyrazole amides as potent inhibitors of the mitotic kinesin KSP
Paul J Coleman, John D Schreier, Christopher D Cox, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 28, 2006
Kinesin spindle protein (KSP) inhibitors. Part 3: synthesis and evaluation of phenolic 2,4-diaryl-2,5-dihydropyrroles with reduced hERG binding and employment of a phosphate prodrug strategy for aqueous solubility
Robert M Garbaccio, Mark E Fraley, Edward S Tasber, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 19, 2006
3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
Mark E Fraley, Justin T Steen, Edward J Brnardic, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 7, 2007
Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors
Edward J Brnardic, Robert M Garbaccio, Mark E Fraley, et al.
Page
of 46
Search research articles
Search
Showing results (431-440 of 459) with videos related to
Sort By:
Page
of 46
Bioorganic & Medicinal Chemistry Letters
|
December 22, 2005
Potent 2-[(pyrimidin-4-yl)amine}-1,3-thiazole-5-carbonitrile-based inhibitors of VEGFR-2 (KDR) kinase
John T Sisko, Thomas J Tucker, Mark T Bilodeau, et al.
Cancer Research
|
December 26, 2001
Evaluation of farnesyl:protein transferase and geranylgeranyl:protein transferase inhibitor combinations in preclinical models
R B Lobell, C A Omer, M T Abrams, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 12, 2001
Non-peptide alpha(v)beta(3) antagonists. Part 3: identification of potent RGD mimetics incorporating novel beta-amino acids as aspartic acid replacements
Paul J Coleman, Karen M Brashear, Cecilia A Hunt, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 28, 2006
Kinesin spindle protein (KSP) inhibitors. Part 2: the design, synthesis, and characterization of 2,4-diaryl-2,5-dihydropyrrole inhibitors of the mitotic kinesin KSP
Mark E Fraley, Robert M Garbaccio, Kenneth L Arrington, et al.
ACS Medicinal Chemistry Letters
|
June 6, 2014
Discovery of 4,4-Disubstituted Quinazolin-2-ones as T-Type Calcium Channel Antagonists
James C Barrow, Kenneth E Rittle, Thomas S Reger, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 30, 2017
Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics
Scott E Wolkenberg, M Brad Nolt, Mark T Bilodeau, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 1, 2007
Kinesin spindle protein (KSP) inhibitors. Part 6: Design and synthesis of 3,5-diaryl-4,5-dihydropyrazole amides as potent inhibitors of the mitotic kinesin KSP
Paul J Coleman, John D Schreier, Christopher D Cox, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 28, 2006
Kinesin spindle protein (KSP) inhibitors. Part 3: synthesis and evaluation of phenolic 2,4-diaryl-2,5-dihydropyrroles with reduced hERG binding and employment of a phosphate prodrug strategy for aqueous solubility
Robert M Garbaccio, Mark E Fraley, Edward S Tasber, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 19, 2006
3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
Mark E Fraley, Justin T Steen, Edward J Brnardic, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 7, 2007
Optimization of a pyrazoloquinolinone class of Chk1 kinase inhibitors
Edward J Brnardic, Robert M Garbaccio, Mark E Fraley, et al.
Page
of 46