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Journal of Medicinal Chemistry|September 27, 2018
Antimalarial Lead-Optimization Studies on a 2,6-Imidazopyridine Series within a Constrained Chemical Space To Circumvent Atypical Dose-Response Curves against Multidrug Resistant Parasite StrainsClaire Le Manach, Tanya Paquet, Kathryn Wicht, et al.ACS Infectious Diseases|December 15, 2020
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and cGMP-Dependent Protein KinasePeter Mubanga Cheuka, Luyanda Centani, Lauren B Arendse, et al.ACS Infectious Diseases|May 30, 2020
Synthesis, Structure-Activity Relationship, and Mechanistic Studies of Aminoquinazolinones Displaying Antimycobacterial ActivityJessica N Akester, Paul Njaria, Aloysius Nchinda, et al.Journal of Medicinal Chemistry|December 12, 2022
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and In Vivo Efficacy in a Plasmodium berghei Mouse Malaria Infection ModelDickson Mambwe, Constance M Korkor, Amanda Mabhula, et al.Journal of Medicinal Chemistry|May 12, 2025
Cell-Based Progression of Spiroindoline Phenotypic Hits Leads to the Identification of Compounds with Diverging Parasitological Profiles against the Human Malaria Parasite Plasmodium falciparumJean Dam, Grant A Boyle, André Horatscheck, et al.Journal of Medicinal Chemistry|June 17, 2021
Benzoheterocyclic Oxime Carbamates Active against Mycobacterium tuberculosis: Synthesis, Structure-Activity Relationship, Metabolism, and Biology TriagingRenier van der Westhuyzen, Amanda Mabhula, Paul M Njaria, et al.Journal of Medicinal Chemistry|February 27, 2014
Medicinal chemistry optimization of antiplasmodial imidazopyridazine hits from high throughput screening of a SoftFocus kinase library: part 1Claire Le Manach, Diego Gonzàlez Cabrera, Frederic Douelle, et al.ACS Infectious Diseases|December 12, 2018
Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of ActionMalkeet Kumar, John Okombo, Dickson Mambwe, et al.Journal of Medicinal Chemistry|October 7, 2025
Optimization of 2,8-Diaryl-1,5-naphthyridines as Plasmodium falciparum Phosphatidylinositol 4-Kinase Inhibitors with Improved ADME Profiles and In Vivo EfficacyGodwin A Dziwornu, Donald Seanego, Stephen Fienberg, et al.Journal of Medicinal Chemistry|April 19, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ null Mouse Model of MalariaAloysius T Nchinda, Claire Le Manach, Tanya Paquet, et al.Pageof 8