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Molecular Pharmaceutics
|
May 12, 2006
Computational models for identifying potential P-glycoprotein substrates and inhibitors
Patrizia Crivori, Benedetta Reinach, Daniele Pezzetta, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences
|
August 24, 2007
Development and validation of in silico models for estimating drug preformulation risk in PEG400/water and Tween80/water systems
Patrizia Crivori, Amedea Morelli, Daniele Pezzetta, et al.
Toxicology in Vitro : an International Journal Published in Association with BIBRA
|
November 25, 2003
Phase I and phase II metabolic activities are retained in liver slices from mouse, rat, dog, monkey and human after cryopreservation
Marcella Martignoni, Mario Monshouwer, Ruben de Kanter, et al.
Xenobiotica; the Fate of Foreign Compounds in Biological Systems
|
March 4, 2015
In vitro and in vivo metabolism of CHF 6001, a selective phosphodiesterase (PDE4) inhibitor
Valentina Cenacchi, Rosangela Battaglia, Flavio Cinato, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 8, 2011
NMS-P937, a 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivative as potent and selective Polo-like kinase 1 inhibitor
Italo Beria, Roberto T Bossi, Maria Gabriella Brasca, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 12, 2010
4,5-Dihydro-1H-pyrazolo[4,3-h]quinazolines as potent and selective Polo-like kinase 1 (PLK1) inhibitors
Italo Beria, Barbara Valsasina, Maria Gabriella Brasca, et al.
Journal of Medicinal Chemistry
|
July 30, 2015
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy
Gianluca Papeo, Helena Posteri, Daniela Borghi, et al.
Journal of Medicinal Chemistry
|
January 1, 2009
First Cdc7 kinase inhibitors: pyrrolopyridinones as potent and orally active antitumor agents. 2. Lead discovery
Maria Menichincheri, Alberto Bargiotti, Jens Berthelsen, et al.
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Search research articles
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Showing results (1-10 of 8) with videos related to
Sort By:
Page
of 1
Molecular Pharmaceutics
|
May 12, 2006
Computational models for identifying potential P-glycoprotein substrates and inhibitors
Patrizia Crivori, Benedetta Reinach, Daniele Pezzetta, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences
|
August 24, 2007
Development and validation of in silico models for estimating drug preformulation risk in PEG400/water and Tween80/water systems
Patrizia Crivori, Amedea Morelli, Daniele Pezzetta, et al.
Toxicology in Vitro : an International Journal Published in Association with BIBRA
|
November 25, 2003
Phase I and phase II metabolic activities are retained in liver slices from mouse, rat, dog, monkey and human after cryopreservation
Marcella Martignoni, Mario Monshouwer, Ruben de Kanter, et al.
Xenobiotica; the Fate of Foreign Compounds in Biological Systems
|
March 4, 2015
In vitro and in vivo metabolism of CHF 6001, a selective phosphodiesterase (PDE4) inhibitor
Valentina Cenacchi, Rosangela Battaglia, Flavio Cinato, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 8, 2011
NMS-P937, a 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivative as potent and selective Polo-like kinase 1 inhibitor
Italo Beria, Roberto T Bossi, Maria Gabriella Brasca, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 12, 2010
4,5-Dihydro-1H-pyrazolo[4,3-h]quinazolines as potent and selective Polo-like kinase 1 (PLK1) inhibitors
Italo Beria, Barbara Valsasina, Maria Gabriella Brasca, et al.
Journal of Medicinal Chemistry
|
July 30, 2015
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy
Gianluca Papeo, Helena Posteri, Daniela Borghi, et al.
Journal of Medicinal Chemistry
|
January 1, 2009
First Cdc7 kinase inhibitors: pyrrolopyridinones as potent and orally active antitumor agents. 2. Lead discovery
Maria Menichincheri, Alberto Bargiotti, Jens Berthelsen, et al.
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