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Drug Discovery Today
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May 8, 2026
Ligand trapping as a key mechanism governing drug residence time, binding affinity, and potency
Danislav S Spassov
International Journal of Molecular Sciences
|
July 13, 2024
Binding Affinity Determination in Drug Design: Insights from Lock and Key, Induced Fit, Conformational Selection, and Inhibitor Trapping Models
Danislav S Spassov
Gene
|
December 3, 2002
Cloning and comparative sequence analysis of PUM1 and PUM2 genes, human members of the Pumilio family of RNA-binding proteins
Danislav S Spassov, Roland Jurecic
Blood Cells, Molecules & Diseases
|
April 2, 2003
Mouse Pum1 and Pum2 genes, members of the Pumilio family of RNA-binding proteins, show differential expression in fetal and adult hematopoietic stem cells and progenitors
Danislav S Spassov, Roland Jurecic
IUBMB Life
|
October 31, 2003
The PUF family of RNA-binding proteins: does evolutionarily conserved structure equal conserved function?
Danislav S Spassov, Roland Jurecic
Molecules (Basel, Switzerland)
|
September 9, 2022
Novel Hits for N-Myristoyltransferase Inhibition Discovered by Docking-Based Screening
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
Frontiers in Molecular Biosciences
|
January 27, 2023
A role of salt bridges in mediating drug potency: A lesson from the N-myristoyltransferase inhibitors
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
International Journal of Molecular Sciences
|
July 29, 2023
Inhibitor Trapping in N-Myristoyltransferases as a Mechanism for Drug Potency
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
International Journal of Molecular Sciences
|
March 28, 2024
Inhibitor Trapping in Kinases
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
Cell Cycle (Georgetown, Tex.)
|
April 15, 2011
Trask phosphorylation defines the reverse mode of a phosphotyrosine signaling switch that underlies cell anchorage state
Danislav S Spassov, Ching H Wong, Mark M Moasser
Page
of 3
Search research articles
Search
Showing results (1-10 of 22) with videos related to
Sort By:
Page
of 3
Drug Discovery Today
|
May 8, 2026
Ligand trapping as a key mechanism governing drug residence time, binding affinity, and potency
Danislav S Spassov
International Journal of Molecular Sciences
|
July 13, 2024
Binding Affinity Determination in Drug Design: Insights from Lock and Key, Induced Fit, Conformational Selection, and Inhibitor Trapping Models
Danislav S Spassov
Gene
|
December 3, 2002
Cloning and comparative sequence analysis of PUM1 and PUM2 genes, human members of the Pumilio family of RNA-binding proteins
Danislav S Spassov, Roland Jurecic
Blood Cells, Molecules & Diseases
|
April 2, 2003
Mouse Pum1 and Pum2 genes, members of the Pumilio family of RNA-binding proteins, show differential expression in fetal and adult hematopoietic stem cells and progenitors
Danislav S Spassov, Roland Jurecic
IUBMB Life
|
October 31, 2003
The PUF family of RNA-binding proteins: does evolutionarily conserved structure equal conserved function?
Danislav S Spassov, Roland Jurecic
Molecules (Basel, Switzerland)
|
September 9, 2022
Novel Hits for N-Myristoyltransferase Inhibition Discovered by Docking-Based Screening
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
Frontiers in Molecular Biosciences
|
January 27, 2023
A role of salt bridges in mediating drug potency: A lesson from the N-myristoyltransferase inhibitors
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
International Journal of Molecular Sciences
|
July 29, 2023
Inhibitor Trapping in N-Myristoyltransferases as a Mechanism for Drug Potency
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
International Journal of Molecular Sciences
|
March 28, 2024
Inhibitor Trapping in Kinases
Danislav S Spassov, Mariyana Atanasova, Irini Doytchinova
Cell Cycle (Georgetown, Tex.)
|
April 15, 2011
Trask phosphorylation defines the reverse mode of a phosphotyrosine signaling switch that underlies cell anchorage state
Danislav S Spassov, Ching H Wong, Mark M Moasser
Page
of 3