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Chemmedchem|February 8, 2014
Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cellsAlessia Lenoci, Stefano Tomassi, Mariarosaria Conte, et al.Chemmedchem|October 25, 2013
Carprofen analogues as sirtuin inhibitors: enzyme and cellular studiesPaolo Mellini, Vincenzo Carafa, Barbara Di Rienzo, et al.ACS Chemical Biology|April 21, 2023
Comparative Study of Adenosine Analogs as Inhibitors of Protein Arginine Methyltransferases and a Clostridioides difficile-Specific DNA Adenine MethyltransferaseJujun Zhou, Youchao Deng, Iredia D Iyamu, et al.Journal of Medicinal Chemistry|February 28, 2017
Development of 1,2,4-Oxadiazoles as Potent and Selective Inhibitors of the Human Deacetylase Sirtuin 2: Structure-Activity Relationship, X-ray Crystal Structure, and Anticancer ActivitySébastien Moniot, Mariantonietta Forgione, Alessia Lucidi, et al.Molecular and Cellular Biology|January 8, 2014
IκB kinase ε targets interferon regulatory factor 1 in activated T lymphocytesMarco Sgarbanti, Giulia Marsili, Anna Lisa Remoli, et al.Plos Currents|September 30, 2010
Evaluation of histone deacetylases as drug targets in Huntington's disease models. Study of HDACs in brain tissues from R6/2 and CAG140 knock-in HD mouse models and human patients and in a neuronal HD cell modelLuisa Quinti, Vanita Chopra, Dante Rotili, et al.Biochemical Pharmacology|January 1, 2016
The histone acetyltransferase p300 inhibitor C646 reduces pro-inflammatory gene expression and inhibits histone deacetylasesThea van den Bosch, Alexander Boichenko, Niek G J Leus, et al.Frontiers in Cell and Developmental Biology|March 13, 2026
Tumor microenvironment-activated ferritin nanovector enables enhanced tumor delivery of KRASG12C inhibitors and degradersAnnalisa Pia Abbinantefina, Claudia Tito, Silvia Masciarelli, et al.International Journal of Molecular Sciences|November 16, 2019
Enzymatic and Biological Characterization of Novel Sirtuin Modulators against CancerVincenzo Carafa, Angelita Poziello, Laura Della Torre, et al.Frontiers in Oncology|June 13, 2020
The Pan-Sirtuin Inhibitor MC2494 Regulates Mitochondrial Function in a Leukemia Cell LineVincenzo Carafa, Rosita Russo, Laura Della Torre, et al.Pageof 20