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Pharmaceuticals (Basel, Switzerland)|February 26, 2022
The Nitrobenzoxadiazole Derivative NBDHEX Behaves as Plasmodium falciparum Gametocyte Selective Inhibitor with Malaria Parasite Transmission Blocking ActivityGiulia Siciliano, Veronica Di Paolo, Dante Rotili, et al.ACS Infectious Diseases|June 22, 2022
Effects of Structurally Different HDAC Inhibitors against Trypanosoma cruzi, Leishmania, and Schistosoma mansoniElisabetta Di Bello, Beatrice Noce, Rossella Fioravanti, et al.Diabetes|October 17, 2012
Inhibition of class I histone deacetylases unveils a mitochondrial signature and enhances oxidative metabolism in skeletal muscle and adipose tissueAndrea Galmozzi, Nico Mitro, Alessandra Ferrari, et al.Journal of Medicinal Chemistry|January 22, 2024
Specific Inhibitors of Mitochondrial Deacylase Sirtuin 4 Endowed with Cellular ActivityMartin Pannek, Zayan Alhalabi, Daniela Tomaselli, et al.European Journal of Medicinal Chemistry|May 21, 2017
The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitorHannah Wapenaar, Thea van den Bosch, Niek G J Leus, et al.Journal of Medicinal Chemistry|March 21, 2012
2-(Alkyl/aryl)amino-6-benzylpyrimidin-4(3H)-ones as inhibitors of wild-type and mutant HIV-1: enantioselectivity studiesDante Rotili, Alberta Samuele, Domenico Tarantino, et al.Journal of Medicinal Chemistry|December 29, 2022
Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile-Specific DNA Adenine Methyltransferase Required for Normal Sporulation and PersistenceJujun Zhou, John R Horton, Martina Menna, et al.Current Radiopharmaceuticals|January 5, 2021
90Y-DOTA-Nimotuzumab: Synthesis of a Promising β- RadiopharmaceuticalTeresa Scotognella, Daria Maccora, Isabella Bruno, et al.International Journal of Molecular Sciences|May 28, 2020
Identification of Inhibitors to Trypanosoma cruzi Sirtuins Based on Compounds Developed to Human EnzymesTanira Matutino Bastos, Milena Botelho Pereira Soares, Caio Haddad Franco, et al.Cell Death & Disease|March 24, 2026
Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemiaGiulia Sgueglia, Crescenzo Massaro, Annamaria Muro, et al.Pageof 20