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European Journal of Medicinal Chemistry|November 20, 2022
Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activityRossella Fioravanti, Eleonora Proia, Ivan N Tyurenkov, et al.Nucleic Acids Research|February 12, 2022
Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcriptionMartina Minisini, Eros Di Giorgio, Emanuela Kerschbamer, et al.Journal of Medicinal Chemistry|July 18, 2008
5-Alkyl-6-benzyl-2-(2-oxo-2-phenylethylsulfanyl)pyrimidin-4(3H)-ones, a series of anti-HIV-1 agents of the dihydro-alkoxy-benzyl-oxopyrimidine family with peculiar structure-activity relationship profileMaxim B Nawrozkij, Dante Rotili, Domenico Tarantino, et al.Biorxiv : the Preprint Server for Biology|March 27, 2026
m 6 A RNA methylation modulates Zika virus infection by regulating serine proteases in Aedes albopictusAnderson de Mendonça Amarante, Lucas Tirloni, Jonas Koch, et al.Cell Chemical Biology|October 22, 2024
Quinoline-based compounds can inhibit diverse enzymes that act on DNAJujun Zhou, Qin Chen, Ren Ren, et al.Journal of Medicinal Chemistry|November 30, 2012
Discovery of salermide-related sirtuin inhibitors: binding mode studies and antiproliferative effects in cancer cells including cancer stem cellsDante Rotili, Domenico Tarantino, Angela Nebbioso, et al.Plos One|May 10, 2014
Properly substituted analogues of BIX-01294 lose inhibition of G9a histone methyltransferase and gain selective anti-DNA methyltransferase 3A activityDante Rotili, Domenico Tarantino, Biagina Marrocco, et al.Journal of Medicinal Chemistry|May 8, 2023
First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8Francesco Fiorentino, Sara Sementilli, Martina Menna, et al.Chemmedchem|February 1, 2020
Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target ModulationRossella Fioravanti, Annalisa Romanelli, Nicola Mautone, et al.Scientific Reports|March 6, 2020
Radioguided surgery with β- radiation in pancreatic Neuroendocrine Tumors: a feasibility studyFrancesco Collamati, Daria Maccora, Sergio Alfieri, et al.Pageof 20