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Clinical Epigenetics|May 27, 2016
Sirtuin functions and modulation: from chemistry to the clinicVincenzo Carafa, Dante Rotili, Mariantonietta Forgione, et al.Journal of Medicinal Chemistry|December 13, 2006
Small-molecule inhibitors of histone acetyltransferase activity: identification and biological propertiesAntonello Mai, Dante Rotili, Domenico Tarantino, et al.Biochemical Pharmacology|June 1, 2020
Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatmentVeronica Di Paolo, Chiara Fulci, Dante Rotili, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|September 29, 2021
Anti-influenza A virus activity and structure-activity relationship of a series of nitrobenzoxadiazole derivativesFrancesco Fiorentino, Marta De Angelis, Martina Menna, et al.Cells|April 23, 2022
Neuroprotective Effects of PARP Inhibitors in Drosophila Models of Alzheimer's DiseaseAnna Maggiore, Assunta Maria Casale, Walter Toscanelli, et al.Journal of Medicinal Chemistry|March 29, 2011
Diarylpyrimidine-dihydrobenzyloxopyrimidine hybrids: new, wide-spectrum anti-HIV-1 agents active at (sub)-nanomolar levelDante Rotili, Domenico Tarantino, Marino Artico, et al.Journal of Molecular Biology|January 10, 2012
An analog of BIX-01294 selectively inhibits a family of histone H3 lysine 9 Jumonji demethylasesAnup K Upadhyay, Dante Rotili, Ji Woong Han, et al.Cancers|February 4, 2021
Regulatory Interplay between miR-181a-5p and Estrogen Receptor Signaling Cascade in Breast CancerRosaria Benedetti, Chiara Papulino, Giulia Sgueglia, et al.Science Advances|September 15, 2016
Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural featuresValentina Speranzini, Dante Rotili, Giuseppe Ciossani, et al.European Journal of Medicinal Chemistry|May 20, 2014
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: enzyme and cellular studiesSimone Carradori, Dante Rotili, Celeste De Monte, et al.Pageof 20