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Scientific Reports|April 27, 2017
The GPR139 reference agonists 1a and 7c, and tryptophan and phenylalanine share a common binding siteAnne Cathrine Nøhr, Willem Jespers, Mohamed A Shehata, et al.ACS Chemical Neuroscience|July 20, 2023
Structure-Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT2A Receptor AgonistsEline Pottie, Christian B M Poulie, Icaro A Simon, et al.Journal of Medicinal Chemistry|September 13, 2022
Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT2A Receptor AgonistsChristian B M Poulie, Eline Pottie, Icaro A Simon, et al.Nature Communications|December 2, 2022
Dynamic spatiotemporal determinants modulate GPCR:G protein coupling selectivity and promiscuityManbir Sandhu, Aaron Cho, Ning Ma, et al.Journal of Medicinal Chemistry|July 13, 2019
Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic LigandsBirgit I Gaiser, Mia Danielsen, Emil Marcher-Rørsted, et al.Trends in Pharmacological Sciences|December 6, 2017
Structural Mapping of Adenosine Receptor Mutations: Ligand Binding and Signaling MechanismsWillem Jespers, Anke C Schiedel, Laura H Heitman, et al.European Journal of Medicinal Chemistry|July 29, 2018
Structure-activity relationship and conformational studies of the natural product cyclic depsipeptides YM-254890 and FR900359Hang Zhang, Alexander L Nielsen, Michael W Boesgaard, et al.Scientific Reports|February 2, 2017
Development of a human vasopressin V1a-receptor antagonist from an evolutionary-related insect neuropeptideMaria Giulia Di Giglio, Markus Muttenthaler, Kasper Harpsøe, et al.Journal of Medicinal Chemistry|February 7, 2023
Comprehensive Peptide Cyclization Examination Yields Optimized APP Scaffolds with Improved Affinity toward Mint2Christian R O Bartling, Flora Alexopoulou, Sarah Kuschert, et al.Molecular Cell|June 17, 2022
GPCRs steer Gi and Gs selectivity via TM5-TM6 switches as revealed by structures of serotonin receptorsSijie Huang, Peiyu Xu, Dan-Dan Shen, et al.Pageof 11