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Bioorganic & Medicinal Chemistry Letters
|
January 16, 2014
Diphenylpyridylethanamine (DPPE)-based aminoheterocycles as cholesteryl ester transfer protein inhibitors
Yufeng Wang, Wu Yang, Heather J Finlay, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 22, 2008
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase
Gretchen M Schroeder, Xiao-Tao Chen, David K Williams, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 22, 2012
Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors
Michael M Miller, Yalei Liu, Ji Jiang, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 1, 2008
2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis
Lalgudi S Harikrishnan, Muthoni G Kamau, Timothy F Herpin, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 2, 2011
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3
Lalgudi S Harikrishnan, Muthoni G Kamau, Honghe Wan, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2008
Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
Haixia Wang, Zheming Ruan, James J Li, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2014
Discovery of pyrrolo[1,2-b]pyridazine-3-carboxamides as Janus kinase (JAK) inhibitors
James J-W Duan, Zhonghui Lu, Bin Jiang, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 26, 2019
Structure based design of macrocyclic factor XIa inhibitors: Discovery of cyclic P1 linker moieties with improved oral bioavailability
Charles G Clark, Karen A Rossi, James R Corte, et al.
Journal of Medicinal Chemistry
|
June 2, 2012
Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors
Lalgudi S Harikrishnan, Heather J Finlay, Jennifer X Qiao, et al.
Journal of Medicinal Chemistry
|
January 24, 2017
Discovery of Pyrrolidine-Containing GPR40 Agonists: Stereochemistry Effects a Change in Binding Mode
Elizabeth A Jurica, Ximao Wu, Kristin N Williams, et al.
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Showing results (11-20 of 20) with videos related to
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Bioorganic & Medicinal Chemistry Letters
|
January 16, 2014
Diphenylpyridylethanamine (DPPE)-based aminoheterocycles as cholesteryl ester transfer protein inhibitors
Yufeng Wang, Wu Yang, Heather J Finlay, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 22, 2008
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase
Gretchen M Schroeder, Xiao-Tao Chen, David K Williams, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 22, 2012
Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors
Michael M Miller, Yalei Liu, Ji Jiang, et al.
Bioorganic & Medicinal Chemistry Letters
|
April 1, 2008
2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis
Lalgudi S Harikrishnan, Muthoni G Kamau, Timothy F Herpin, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 2, 2011
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3
Lalgudi S Harikrishnan, Muthoni G Kamau, Honghe Wan, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2008
Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
Haixia Wang, Zheming Ruan, James J Li, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 3, 2014
Discovery of pyrrolo[1,2-b]pyridazine-3-carboxamides as Janus kinase (JAK) inhibitors
James J-W Duan, Zhonghui Lu, Bin Jiang, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 26, 2019
Structure based design of macrocyclic factor XIa inhibitors: Discovery of cyclic P1 linker moieties with improved oral bioavailability
Charles G Clark, Karen A Rossi, James R Corte, et al.
Journal of Medicinal Chemistry
|
June 2, 2012
Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors
Lalgudi S Harikrishnan, Heather J Finlay, Jennifer X Qiao, et al.
Journal of Medicinal Chemistry
|
January 24, 2017
Discovery of Pyrrolidine-Containing GPR40 Agonists: Stereochemistry Effects a Change in Binding Mode
Elizabeth A Jurica, Ximao Wu, Kristin N Williams, et al.
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